Mebufotenin

Mebufotenin

SCHEMBL25344818

O=C(O)/C=C/C(=O)O.[2H]C([2H])(Cc1c[nH]c2ccc(OC)cc12)N(C)C

nearest known ligand 0.68

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ADRB1ADRB2ATP4AATP4BAXLCHRM2CHRM3DRD2FLT3HRH1HTR2AHTR2BHTR2CKCNH2KMT2AMAP2K1MAP2K2MEN1MLNRPLK4RENS1PR1SLC6A2SLC6A4atpAatpBatpCatpDatpEatpFatpFHatpGpol

The experimentally established mechanism targets of Mebufotenin. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2B known ✓ P41595 4/20 0.68
HTR2A known ✓ P28223 4/20 0.68
HTR2C known ✓ P28335 4/20 0.68
HRH1 known ✓ P35367 2/20 0.68
KMT2A known ✓ Q03164 2/20 0.67
SLC6A4 known ✓ P31645 2/20 0.59
MEN1 known ✓ O00255 1/20 0.56
SLC6A2 known ✓ P23975 1/20 0.55
HTR1A P08908 6/20 0.68
HTR1B P28222 6/20 0.68
HTR7 P34969 4/20 0.68
HTR6 P50406 4/20 0.68
HTR5A P47898 3/20 0.68
ADRA2A P08913 2/20 0.68
ADRA2B P18089 2/20 0.68
ADRA2C P18825 2/20 0.68
MAOA P21397 1/20 0.68
ADRA1D P25100 1/20 0.68
CHRNB4 P30926 1/20 0.68
CHRNA3 P32297 1/20 0.68

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Mebufotenin SCHEMBL30777166 0.89 HTR2A (0.75) HTR1AHTR1BHTR2BHTR2AHTR2C
Mebufotenin SCHEMBL25418408 0.89 HTR2A (0.75) HTR1AHTR1BHTR2BHTR2AHTR2C
Mebufotenin SCHEMBL30199593 0.89 KMT2A (0.84) HTR1AHTR1BHTR2BHTR2AHTR2C
Mebufotenin SCHEMBL23927938 0.89 KMT2A (0.84) HTR1AHTR1BHTR2BHTR2AHTR2C
5-Methoxytryptamine SCHEMBL30933118 0.84 HTR1A (0.78) HTR1AHTR1BHTR2BHTR2AHTR2C
5-Methoxytryptamine SCHEMBL31240192 0.84 HTR1A (0.78) HTR1AHTR1BHTR2BHTR2AHTR2C
5-Methoxytryptamine SCHEMBL7094587 0.84 HTR1A (0.78) HTR1AHTR1BHTR2BHTR2AHTR2C
5-Methoxytryptamine SCHEMBL7094589 0.84 HTR1A (0.78) HTR1AHTR1BHTR2BHTR2AHTR2C
5-Methoxytryptamine SCHEMBL30960099 0.83 HTR1A (0.76) HTR1AHTR1BHTR2BHTR2AHTR2C
Mebufotenin SCHEMBL25184829 0.82 HTR2A (0.67) HTR1AHTR1BHTR2BHTR2AHTR2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230250059-A1 SYNTHESIS OF N,N-DIMETHYLTRYPTAMINE-TYPE COMPOUNDS, METHODS, AND USES SMALL PHARMA LTD (GB) 2023-08-10 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230250059-A1 SYNTHESIS OF N,N-DIMETHYLTRYPTAMINE-TYPE COMPOUNDS, METHODS, AND USES TPH2, TPH1, HTR2C HTR2B 17/4885HTR2A 9/4885HTR2C 3/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.