SCHEMBL25345484

SCHEMBL25345484

Cc1nc(C)c(CC(CCCC(=O)O)(C(=O)O)c2ccccn2)nc1C

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BLM P54132 2/20 0.38
CYP2D6 P10635 1/20 0.38
SMN1; SMN2 Q16637 3/20 0.36
APP P05067 1/20 0.35
ALDH1A1 P00352 2/20 0.34
TBXA2R P21731 2/20 0.34
HTT P42858 2/20 0.33
LMNA P02545 1/20 0.33
SLC22A2 O15244 1/20 0.33
SLC22A1 O15245 1/20 0.33
PGR P06401 1/20 0.33
THRB P10828 1/20 0.33
ADRB3 P13945 1/20 0.33
OPRK1 P41145 1/20 0.33
PMP22 Q01453 1/20 0.33
KCNH2 Q12809 1/20 0.33
PDE3A Q14432 1/20 0.33
SLC47A1 Q96FL8 1/20 0.33
CYP3A4 P08684 1/20 0.33
ALOX15 P16050 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25344083 0.87 BLM (0.35) BLMCYP2D6SMN1; SMN2APPTBXA2R
SCHEMBL25345205 0.79 L3MBTL1 (0.38) BLMCYP2D6SMN1; SMN2APPALDH1A1
SCHEMBL4861916 0.70 BLM (0.46) BLMCYP2D6SMN1; SMN2ALDH1A1TBXA2R
SCHEMBL6532232 0.65 SMN1; SMN2 (0.42) BLMCYP2D6SMN1; SMN2ALDH1A1HTT
SCHEMBL1697473 0.64 BLM (0.48) BLMCYP2D6SMN1; SMN2ALDH1A1TBXA2R
SCHEMBL28186562 0.64 SMN1; SMN2 (0.41) BLMCYP2D6SMN1; SMN2ALDH1A1HTT
Ligustrazine SCHEMBL28678860 0.63 LMNA (0.58) APPALDH1A1LMNAPMP22PDE3A
SCHEMBL7315392 0.62 BLM (0.41) BLMCYP2D6SMN1; SMN2ALDH1A1TBXA2R
SCHEMBL505194 0.61 L3MBTL1 (0.52) BLMCYP2D6SMN1; SMN2ALDH1A1LMNA
SCHEMBL5074249 0.61 L3MBTL1 (0.52) BLMCYP2D6SMN1; SMN2ALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023134682-A1 OPTICALLY ACTIVE 2-HYDROXYTETRAHYDROTHIENOPYRIDINE DERIVATIVE, AND PREPARATION METHOD THEREFOR AND USE THEREOF 天地恒一制药股份有限公司 2023-07-20 WO disclosed