SCHEMBL25398564

SCHEMBL25398564

O=[N+]([O-])c1ccc(OCCN2CCSCC2)nc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.50
LTA4H P09960 3/20 0.48
PTGS2 P35354 2/20 0.48
PTGS1 P23219 1/20 0.48
ALDH1A1 P00352 5/20 0.45
TDP1 Q9NUW8 2/20 0.45
LMNA P02545 2/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
MAPT P10636 5/20 0.44
HRH3 Q9Y5N1 1/20 0.42
HSPB1 P04792 1/20 0.42
ALOX12 P18054 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
KCNJ1 P48048 1/20 0.40
KCNH2 Q12809 1/20 0.40
DPP4 P27487 1/20 0.40
GAA P10253 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
CYP1A2 P05177 1/20 0.39
CYP2C9 P11712 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1641137 0.88 LTA4H (0.61) KDM4ELTA4HPTGS2PTGS1ALDH1A1
SCHEMBL6408582 0.87 LTA4H (0.60) KDM4ELTA4HPTGS2PTGS1ALDH1A1
SCHEMBL3382465 0.86 ALDH1A1 (0.49) KDM4ELTA4HPTGS2PTGS1ALDH1A1
SCHEMBL3386044 0.85 ALDH1A1 (0.54) KDM4ELTA4HPTGS2PTGS1ALDH1A1
SCHEMBL16973009 0.82 LTA4H (0.46) KDM4ELTA4HPTGS2PTGS1ALDH1A1
SCHEMBL22171219 0.82 MAPT (0.56) KDM4ELTA4HPTGS2PTGS1ALDH1A1
SCHEMBL6643718 0.79 CYP1A2 (0.59) KDM4EALDH1A1LMNASMN1; SMN2MAPT
SCHEMBL25399700 0.77 LTA4H (0.46) KDM4ELTA4HPTGS2PTGS1MAPT
SCHEMBL13736688 0.77 CD38 (0.41) KDM4ELTA4HPTGS2PTGS1ALDH1A1
SCHEMBL25398475 0.76 ALDH1A1 (0.55) KDM4ELTA4HPTGS2PTGS1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023177356-A2 COMPOUNDS AND METHOD FOR PKMYT1 INHIBITION ENGINE BIOSCIENCES PTE. LTD. (SG) 2023-09-21 WO disclosed