SCHEMBL25399545

SCHEMBL25399545

COc1csc(C(N)=O)c1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 5/20 0.54
MEN1 O00255 3/20 0.54
HTT P42858 2/20 0.45
HPGD P15428 1/20 0.45
PARP1 P09874 2/20 0.44
PARP10 Q53GL7 2/20 0.44
CA1 P00915 1/20 0.44
CA2 P00918 1/20 0.44
PARP2 Q9UGN5 1/20 0.44
PARP4 Q9UKK3 1/20 0.44
CDK2 P24941 1/20 0.42
IKBKE Q14164 1/20 0.42
AURKB Q96GD4 1/20 0.42
TBK1 Q9UHD2 1/20 0.42
IKBKB O14920 1/20 0.39
ICAM1 P05362 2/20 0.39
SELE P16581 2/20 0.39
MAPT P10636 1/20 0.39
CCNC P24863 1/20 0.38
CDK8 P49336 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28147113 0.83 MEN1 (0.39) KMT2AMEN1HTTCA2MAPT
SCHEMBL4703482 0.82 DAO (0.55) KMT2AMEN1HPGDCA1CA2
SCHEMBL18302448 0.82 MAPT (0.52) KMT2AMEN1HPGDIKBKEAURKB
SCHEMBL25399448 0.80 OPRD1 (0.45) KMT2AMEN1HPGDCA1CA2
SCHEMBL3055932 0.80 MEN1 (0.37) KMT2AMEN1HPGDCA2MAPT
Hydrochloric Acid SCHEMBL30515341 0.78 MEN1 (0.37) KMT2AMEN1CA2MAPTMAPK1
SCHEMBL28148274 0.77 KMT2A (0.43) KMT2AMEN1MAPTNPSR1
SCHEMBL24579380 0.77 ALDH1A1 (0.38) KMT2AMEN1CA1CA2MAPT
SCHEMBL6870004 0.76 HSD17B1 (0.64) HTTHPGDPARP1CDK2IKBKE
SCHEMBL8632472 0.75 MAPT (0.39) KMT2AMEN1CA1CA2AURKB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230365584-A1 HETEROCYCLIC PERICONDENSED CDC7 KINASE INHIBITORS FOR THE TREATMENT OF CANCER SCHRÖDINGER, INC. 2023-11-16 US disclosed
US-20230365584-A1 HETEROCYCLIC PERICONDENSED CDC7 KINASE INHIBITORS FOR THE TREATMENT OF CANCER SCHRÖDINGER, INC. 2023-11-16 US disclosed
US-20230365584-A1 HETEROCYCLIC PERICONDENSED CDC7 KINASE INHIBITORS FOR THE TREATMENT OF CANCER SCHRÖDINGER, INC. 2023-11-16 US disclosed
CN-116490507-A Heterocyclic condensation CDC7 kinase inhibitors for the treatment of cancer 薛定谔公司 2023-07-25 CN disclosed
EP-4211140-A1 HETEROCYCLIC PERICONDENSED CDC7 KINASE INHIBITORS FOR THE TREATMENT OF CANCER Schrödinger, Inc. (US) 2023-07-19 EP disclosed
WO-2022055963-A1 HETEROCYCLIC PERICONDENSED CDC7 KINASE INHIBITORS FOR THE TREATMENT OF CANCER SCHRÖDINGER, INC. (US) 2022-03-17 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230365584-A1 HETEROCYCLIC PERICONDENSED CDC7 KINASE INHIBITORS FOR THE TREATMENT OF CANCER CDC7, BUB1B, CDK7 KMT2A 1874/4885MEN1 1575/4885HTT 4640/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.