SCHEMBL25401830

SCHEMBL25401830

COC(=O)c1ccc2cn(Cc3cccnc3)nc2c1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 1/20 0.50
CYP11B1 P15538 1/20 0.50
CYP11B2 P19099 1/20 0.50
KDM4E B2RXH2 1/20 0.47
ALDH1A1 P00352 2/20 0.46
EGFR P00533 1/20 0.46
MAPK1 P28482 2/20 0.45
TSHR P16473 1/20 0.45
ALOX15 P16050 1/20 0.43
HTT P42858 1/20 0.43
TP53 P04637 3/20 0.43
SMN1; SMN2 Q16637 3/20 0.43
CYP3A4 P08684 2/20 0.43
TDP1 Q9NUW8 1/20 0.43
POLB P06746 2/20 0.42
MAPT P10636 2/20 0.42
KDM4C Q9H3R0 1/20 0.42
IRAK4 Q9NWZ3 1/20 0.42
USP2 O75604 1/20 0.42
NPSR1 Q6W5P4 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30584939 1.00 CYP19A1 (0.50) CYP19A1CYP11B1CYP11B2KDM4EALDH1A1
SCHEMBL5767415 0.87 P2RX7 (0.48) ALDH1A1TSHRTP53MAPTGAA
SCHEMBL25402399 0.86 L3MBTL1 (0.48) ALDH1A1HTTTDP1POLBKDM4C
SCHEMBL30585030 0.85 HDAC6 (0.51) ALDH1A1
SCHEMBL25399686 0.85 HDAC6 (0.51) ALDH1A1
SCHEMBL25403016 0.82 MRGPRX4 (0.46) KDM4EALDH1A1MAPK1SMN1; SMN2MAPT
SCHEMBL25399737 0.82 CD74 (0.48) MAPT
SCHEMBL25401651 0.82 THRB (0.53) KDM4ETP53MAPTKLKB1
SCHEMBL25403100 0.82 POLB (0.46) KDM4EALDH1A1ALOX15HTTPOLB
SCHEMBL25402366 0.81 HDAC6 (0.49) SMN1; SMN2MAPTNPSR1KLKB1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023177250-A1 NOVEL HETEROCYCLIC INHIBITOR FOR HISTONE DEACETYLASE, AND PHARMACEUTICAL COMPOSITION COMPRISING SAME 숙명여자대학교산학협력단 2023-09-21 WO disclosed