SCHEMBL254164

SCHEMBL254164

COC(=O)[C@@H](NC(=O)c1ccc(-c2ccc(N)cc2)cc1)C(C)(C)NC(=O)OC(C)(C)C

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.36
RAB9A P51151 1/20 0.36
CA2 P00918 2/20 0.35
ESRRG P62508 1/20 0.35
CA12 O43570 1/20 0.34
CA1 P00915 1/20 0.34
CA9 Q16790 1/20 0.34
CA14 Q9ULX7 1/20 0.34
ADRB2 P07550 1/20 0.34
ADRB1 P08588 1/20 0.34
ADRB3 P13945 1/20 0.34
CYP17A1 P05093 1/20 0.34
DRD2 P14416 1/20 0.34
DRD3 P35462 1/20 0.34
EPHX2 P34913 1/20 0.34
ALDH1A1 P00352 1/20 0.34
CYP3A4 P08684 1/20 0.34
CYP26A1 O43174 1/20 0.34
HDAC1 Q13547 1/20 0.34
CD274 Q9NZQ7 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20299909 0.90 ACACB (0.36) NPC1RAB9ACA2ADRB2ADRB1
SCHEMBL13984819 0.89 MIF (0.37) CA2CA12CA1CA9CA14
SCHEMBL15235730 0.88 ADRB2 (0.34) NPC1RAB9ACA2ESRRGADRB2
SCHEMBL13267033 0.86 GPR119 (0.40) ADRB2ADRB1ADRB3CYP17A1EPHX2
SCHEMBL16820663 0.84 TAS1R3 (0.35) CA2TAS1R3TAS1R1
SCHEMBL30479489 0.84 ALDH1A1 (0.43) NPC1RAB9ACA12CA14ALDH1A1
SCHEMBL30479490 0.84 ALDH1A1 (0.43) NPC1RAB9ACA12CA14ALDH1A1
SCHEMBL16820664 0.84 TAS1R3 (0.35) CA2TAS1R3TAS1R1
SCHEMBL13984789 0.83 PPARA (0.41) RAB9AALDH1A1HDAC1TAS1R3TAS1R1
SCHEMBL13267265 0.82 ALDH1A1 (0.49) ALDH1A1TAS1R3TAS1R1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012031298-A2 ETHYNYLBENZENE DERIVATIVES DUKE UNIVERSITY (US) 2012-03-08 WO disclosed