SCHEMBL25417152

SCHEMBL25417152

O=c1ccc(-c2nc(-c3cncc(Cl)c3)no2)n[nH]1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 7/20 0.45
TP53 P04637 5/20 0.45
FGFR1 P11362 1/20 0.37
CYP1A2 P05177 1/20 0.37
NPC1 O15118 3/20 0.37
KDM4E B2RXH2 1/20 0.37
HPGD P15428 1/20 0.37
HSD17B10 Q99714 1/20 0.37
GPR119 Q8TDV5 1/20 0.36
CASP3 P42574 2/20 0.36
RAB9A P51151 2/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
PRMT5 O14744 1/20 0.36
WDR77 Q9BQA1 1/20 0.36
POLB P06746 1/20 0.36
MEN1 O00255 1/20 0.35
LMNA P02545 1/20 0.35
KMT2A Q03164 1/20 0.35
MKNK1 Q9BUB5 1/20 0.35
MKNK2 Q9HBH9 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31150586 1.00 MAPT (0.45) MAPTTP53FGFR1CYP1A2NPC1
SCHEMBL25418543 0.84 MAPT (0.63) MAPTTP53NPC1RAB9AL3MBTL1
SCHEMBL30419948 0.84 MAPT (0.63) MAPTTP53NPC1RAB9AL3MBTL1
SCHEMBL25189026 0.72 KMT2A (0.39) FGFR1CYP1A2NPC1KDM4ERAB9A
SCHEMBL24783657 0.72 LMNA (0.65) MAPTTP53NPC1KDM4EHPGD
SCHEMBL24038686 0.71 MET (0.46) TP53POLBMEN1KMT2A
SCHEMBL3216138 0.69 LMNA (0.49) MAPTTP53CYP1A2GPR119POLB
SCHEMBL15505029 0.69 MAPT (0.47) MAPTTP53CYP1A2NPC1HPGD
SCHEMBL14881124 0.69 CASP3 (0.56) MAPTTP53CASP3L3MBTL1POLB
SCHEMBL14884856 0.68 NPC1 (0.45) MAPTTP53NPC1KDM4EHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4433473-A1 PYRIDAZINONE COMPOUNDS AND USES THEREOF EDGEWISE THERAPEUTICS, INC. (US) 2024-09-25 EP disclosed
WO-2023091606-A1 PYRIDAZINONE COMPOUNDS AND USES THEREOF EDGEWISE THERAPEUTICS, INC. (US) 2023-05-25 WO disclosed
WO-2023091606-A1 PYRIDAZINONE COMPOUNDS AND USES THEREOF EDGEWISE THERAPEUTICS, INC. (US) 2023-05-25 WO disclosed