SCHEMBL25428534

SCHEMBL25428534

C[C@@H]1Cc2ncc(C#N)cc2CN1C(=O)O

nearest known ligand 0.36

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 4/20 0.36
EGLN2 Q96KS0 1/20 0.34
PDK1 Q15118 3/20 0.33
PDK2 Q15119 3/20 0.33
GRM5 P41594 3/20 0.32
P2RX7 Q99572 1/20 0.32
SSTR4 P31391 1/20 0.32
HCRTR2 O43614 2/20 0.32
HCRTR1 O43613 1/20 0.32
RIPK1 Q13546 1/20 0.32
FNTA P49354 2/20 0.32
FNTB P49356 2/20 0.32
SCD5 Q86SK9 1/20 0.31
EGLN1 Q9GZT9 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25428538 1.00 BRD4 (0.36) BRD4EGLN2PDK1PDK2GRM5
SCHEMBL26026395 0.84 GPR119 (0.40) EGLN2SSTR4
SCHEMBL23326979 0.81 P2RX7 (0.33) GRM5P2RX7
SCHEMBL25429344 0.80 ABHD6 (0.41)
SCHEMBL25431503 0.80 ABHD6 (0.41)
SCHEMBL25428247 0.80 OPRM1 (0.31) PDK1PDK2
SCHEMBL25428241 0.80 OPRM1 (0.31) PDK1PDK2
SCHEMBL25427523 0.76 ROCK1 (0.35)
SCHEMBL25427529 0.76 ROCK1 (0.35)
SCHEMBL23327016 0.73 ELANE (0.35)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023154282-A1 COMPOUNDS HAVING A T-STRUCTURE FORMED BY AT LEAST FOUR CYCLES FOR USE IN THE TREATMENT OF CANCER AND OTHER INDICATIONS THERAS, INC. (US) 2023-08-17 WO disclosed