Splitomicin

Splitomicin

SCHEMBL2544804

O=C1CCc2c(ccc3ccccc23)O1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
SIRT1 Q96EB6 2/20 1.00
KDM4E B2RXH2 1/20 1.00
CYP1A2 P05177 1/20 1.00
GLA P06280 1/20 1.00
CYP2C9 P11712 1/20 1.00
HPGD P15428 1/20 1.00
CYP2C19 P33261 1/20 1.00
HSD17B10 Q99714 1/20 1.00
SIRT2 Q8IXJ6 3/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Splitomicin SCHEMBL29570541 1.00 SIRT1 (1.00) SIRT1KDM4ECYP1A2GLACYP2C9
SCHEMBL13893535 0.90 SIRT1 (0.81) SIRT1KDM4ECYP1A2GLACYP2C9
SCHEMBL14677465 0.84 SIRT1 (0.72) SIRT1KDM4ECYP1A2GLACYP2C9
SCHEMBL13893534 0.79 KDM4E (0.65) SIRT1KDM4ECYP1A2GLACYP2C9
SCHEMBL9121753 0.78 HPGD (0.64) SIRT1KDM4ECYP1A2GLACYP2C9
SCHEMBL9123291 0.78 HPGD (0.64) SIRT1KDM4ECYP1A2GLACYP2C9
SCHEMBL8313602 0.75 KDM4E (0.60) SIRT1KDM4ECYP1A2GLACYP2C9
SCHEMBL30522627 0.75 KDM4E (0.60) SIRT1KDM4ECYP1A2GLACYP2C9
SCHEMBL414928 0.75 HSD17B10 (0.59) SIRT1KDM4ECYP1A2GLACYP2C9
SCHEMBL29688038 0.75 HSD17B10 (0.59) SIRT1KDM4ECYP1A2GLACYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 75 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20220378782-A1 KCC2 EXPRESSION ENHANCING COMPOUNDS AND USES THEREOF WHITEHEAD INSTITUTE FOR BIOMEDICAL RESEARCH (US) 2022-12-01 US claimed
US-9168316-B2 Methods for treating obesity GU YANSONG (US) 2015-10-27 US claimed
US-20140322136-A1 METHODS FOR TREATING OBESITY GU YANSONG (US) 2014-10-30 US claimed
US-20110262362-A1 METHODS FOR TREATING OBESITY GU YANSONG 2011-10-27 US claimed
WO-2010042868-A2 METHODS FOR TREATING OBESITY UNIVERSITY OF WASHINGTON (US) 2010-04-15 WO claimed
US-20060194769-A1 Small molecules that reduce fungal growth UNIVERSITY OF VERMONT AND STATE AGRICULTURAL COLLEGE (US) 2006-08-31 US claimed
WO-2006081327-A2 SMALL MOLECULES THAT REDUCE FUNGAL GROWTH UNIVERSITY OF VERMONT AND STATE AGRICULTURAL COLLEGE (US) 2006-08-03 WO claimed
US-20050079995-A1 Methods for inhibiting deacetylase activity NATIONAL INSTITUTES OF HEALTH - DIRECTOR DEITR 2005-04-14 US claimed
WO-2003046207-A2 METHODS FOR INHIBITING DEACETYLASE ACTIVITY FRED HUTCHINSON CANCER RESEARCH CENTER (US) 2003-06-05 WO claimed
EP-4194548-B1 GENERATION OF HUMAN PLURIPOTENT STEM CELL DERIVED FUNCTIONAL BETA CELLS SHOWING A GLUCOSE-DEPENDENT MITOCHONDRIAL RESPIRATION AND TWO-PHASE INSULIN SECRETION RESPONSE JANSSEN BIOTECH INC (US) 2025-10-22 EP disclosed
US-12408605-B2 Haploid embryogenesis STICHTING WAGENINGEN RESEARCH (NL) 2025-09-09 US disclosed
US-20250218546-A1 METHODS AND COMPOSITIONS FOR SIRT1 EXPRESSION AS A MARKER FOR ENDOMETRIOSIS AND SUBFERTILITY Prisma Health 2025-07-03 US disclosed
US-20240100079-A1 METHODS AND COMPOSITIONS FOR REGENERATING HAIR CELLS IN THE INNER EAR OF ADULT MAMMALS NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2024-03-28 US disclosed
EP-4288066-A1 METHODS AND COMPOSITIONS FOR REGENERATING HAIR CELLS IN THE INNER EAR OF ADULT MAMMALS Massachusetts Eye and Ear Infirmary (US) 2023-12-13 EP disclosed
WO-2006081327-A2 SMALL MOLECULES THAT REDUCE FUNGAL GROWTH UNIVERSITY OF VERMONT AND STATE AGRICULTURAL COLLEGE (US) 2006-08-03 WO disclosed
WO-2006081327-A2 SMALL MOLECULES THAT REDUCE FUNGAL GROWTH UNIVERSITY OF VERMONT AND STATE AGRICULTURAL COLLEGE (US) 2006-08-03 WO disclosed
US-20050079995-A1 Methods for inhibiting deacetylase activity NATIONAL INSTITUTES OF HEALTH - DIRECTOR DEITR 2005-04-14 US disclosed
WO-2003046207-A2 METHODS FOR INHIBITING DEACETYLASE ACTIVITY FRED HUTCHINSON CANCER RESEARCH CENTER (US) 2003-06-05 WO disclosed
WO-2003046207-A2 METHODS FOR INHIBITING DEACETYLASE ACTIVITY FRED HUTCHINSON CANCER RESEARCH CENTER (US) 2003-06-05 WO disclosed
WO-1997014685-A1 PYRIMIDINE DERIVATIVES GYÓGYSZERKUTATÓ INTÉZET KFT (HU) 1997-04-24 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060194769-A1 Small molecules that reduce fungal growth ERG28, DPM1, CYP51A1 SIRT1 2725/4885KDM4E 2135/4885CYP1A2 1362/4885
US-20220378782-A1 KCC2 EXPRESSION ENHANCING COMPOUNDS AND USES THEREOF MECP2, SLC1A2, GRIN2C SIRT1 4028/4885KDM4E 127/4885CYP1A2 4732/4885
US-20050079995-A1 Methods for inhibiting deacetylase activity SIRT2, SIRT1, HDAC1 SIRT1 2/4885KDM4E 1476/4885CYP1A2 4122/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.