Splitomicin

Splitomicin

SCHEMBL29570541

O=C1CCc2c(ccc3ccccc23)O1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
SIRT1 Q96EB6 2/20 1.00
KDM4E B2RXH2 1/20 1.00
CYP1A2 P05177 1/20 1.00
GLA P06280 1/20 1.00
CYP2C9 P11712 1/20 1.00
HPGD P15428 1/20 1.00
CYP2C19 P33261 1/20 1.00
HSD17B10 Q99714 1/20 1.00
SIRT2 Q8IXJ6 3/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Splitomicin SCHEMBL2544804 1.00 SIRT1 (1.00) SIRT1KDM4ECYP1A2GLACYP2C9
SCHEMBL13893535 0.90 SIRT1 (0.81) SIRT1KDM4ECYP1A2GLACYP2C9
SCHEMBL14677465 0.84 SIRT1 (0.72) SIRT1KDM4ECYP1A2GLACYP2C9
SCHEMBL13893534 0.79 KDM4E (0.65) SIRT1KDM4ECYP1A2GLACYP2C9
SCHEMBL9121753 0.78 HPGD (0.64) SIRT1KDM4ECYP1A2GLACYP2C9
SCHEMBL9123291 0.78 HPGD (0.64) SIRT1KDM4ECYP1A2GLACYP2C9
SCHEMBL8313602 0.75 KDM4E (0.60) SIRT1KDM4ECYP1A2GLACYP2C9
SCHEMBL30522627 0.75 KDM4E (0.60) SIRT1KDM4ECYP1A2GLACYP2C9
SCHEMBL414928 0.75 HSD17B10 (0.59) SIRT1KDM4ECYP1A2GLACYP2C9
SCHEMBL29688038 0.75 HSD17B10 (0.59) SIRT1KDM4ECYP1A2GLACYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 35 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3841097-B1 2,6-BIS(((1H-BENZO[D]IMIDAZOL-2-YL)THIO)METHYL)PYRIDINE AND N2,N6-DIBENZYLPYRIDINE-2,6-DICARBOXAMIDE DERIVATIVES AND RELATED COMPOUNDS AS PHOSPHOINOSITIDE 3-KINASE (PI3K) INHIBITORS FOR TREATING CANCER BIOMEDICAL RES FOUNDATION OF THE ACADEMY OF ATHENS BRFAA (GR) 2026-05-20 EP claimed
US-12496357-B2 Compositions and methods for treating sickle cell disease YALE UNIVERSITY (US) 2025-12-16 US claimed
WO-2024192348-A2 METHODS OF TREATING HPV IN HIV-INFECTED PATIENTS OHIO STATE INNOVATION FOUNDATION (US) 2024-09-19 WO claimed
US-20220280656-A1 COMPOSITIONS AND METHODS FOR TREATING SICKLE CELL DISEASE YALE UNIVERSITY 2022-09-08 US claimed
US-20220249477-A1 METHODS AND COMPOSITIONS FOR TREATING VIRAL OR VIRALLY-INDUCED CONDITIONS VIRACTA THERAPEUTICS, INC. (US) 2022-08-11 US claimed
EP-3319965-B1 NOVEL COMPOUNDS FOR USE IN TREATING OR PREVENTING CANCEROUS DISEASES BIOMEDICAL RES FOUNDATION OF THE ACADEMY OF ATHENS (GR) 2022-05-04 EP claimed
EP-3841097-B1 2,6-BIS(((1H-BENZO[D]IMIDAZOL-2-YL)THIO)METHYL)PYRIDINE AND N2,N6-DIBENZYLPYRIDINE-2,6-DICARBOXAMIDE DERIVATIVES AND RELATED COMPOUNDS AS PHOSPHOINOSITIDE 3-KINASE (PI3K) INHIBITORS FOR TREATING CANCER BIOMEDICAL RES FOUNDATION OF THE ACADEMY OF ATHENS BRFAA (GR) 2026-05-20 EP disclosed
EP-4715066-A1 PANEL OF MICRORNAS AS BIOMARKERS OF NON-SEGMENTAL VITILIGO Servicio Andaluz De Salud (ES) 2026-03-25 EP disclosed
EP-4691479-A2 GENERATION OF HUMAN PLURIPOTENT STEM CELL DERIVED FUNCTIONAL BETA CELLS SHOWING A GLUCOSE-DEPENDENT MITOCHONDRIAL RESPIRATION AND TWO-PHASE INSULIN SECRETION RESPONSE Janssen Biotech, Inc. (US) 2026-02-11 EP disclosed
US-12496357-B2 Compositions and methods for treating sickle cell disease YALE UNIVERSITY (US) 2025-12-16 US disclosed
US-20250281445-A1 Method of dietary treatment for genetic and epigenetic diseases and disorders OTT DAVID MICHAEL (US) 2025-09-11 US disclosed
US-12338198-B2 Cancer cell growth inhibiting composition and processed food Hagihara Farm Production Institute Co., Ltd. (JP) 2025-06-24 US disclosed
US-20240390375-A1 METHODS AND COMPOSITIONS FOR TREATING VIRAL OR VIRALLY-INDUCED CONDITIONS Viracta Subsidiary, Inc. (US) 2024-11-28 US disclosed
US-20220378782-A1 KCC2 EXPRESSION ENHANCING COMPOUNDS AND USES THEREOF WHITEHEAD INSTITUTE FOR BIOMEDICAL RESEARCH (US) 2022-12-01 US disclosed
US-20220280656-A1 COMPOSITIONS AND METHODS FOR TREATING SICKLE CELL DISEASE YALE UNIVERSITY 2022-09-08 US disclosed
US-20220249477-A1 METHODS AND COMPOSITIONS FOR TREATING VIRAL OR VIRALLY-INDUCED CONDITIONS VIRACTA THERAPEUTICS, INC. (US) 2022-08-11 US disclosed
WO-2022115581-A1 METHODS FOR TREATING INFERTILITY AND/OR ENDOMETRIOSIS COMPRISING EX-527 THE UNIVERSITY OF NORTH CAROLINA AT CHAPEL HILL (US) 2022-06-02 WO disclosed
US-11331313-B2 KCC2 expression enhancing compounds and uses thereof WHITEHEAD INSTITUTE FOR BIOMEDICAL RESEARCH (US) 2022-05-17 US disclosed
US-20220135514-A1 CANCER CELL GROWTH INHIBITING COMPOSITION AND PROCESSED FOOD Hagihara Farm Production Institute Co., Ltd. (JP) 2022-05-05 US disclosed
EP-3319965-B1 NOVEL COMPOUNDS FOR USE IN TREATING OR PREVENTING CANCEROUS DISEASES BIOMEDICAL RES FOUNDATION OF THE ACADEMY OF ATHENS (GR) 2022-05-04 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (6 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11331313-B2 KCC2 expression enhancing compounds and uses thereof MECP2, SLC1A2, GRIN2C SIRT1 4028/4885KDM4E 127/4885CYP1A2 4732/4885
US-12338198-B2 Cancer cell growth inhibiting composition and processed food MKI67, FLOT1, VHL SIRT1 4483/4885KDM4E 3370/4885CYP1A2 3310/4885
US-20220280656-A1 COMPOSITIONS AND METHODS FOR TREATING SICKLE CELL DISEASE HBB, HBG1, HBZ SIRT1 4760/4885KDM4E 4884/4885CYP1A2 4657/4885
US-20220135514-A1 CANCER CELL GROWTH INHIBITING COMPOSITION AND PROCESSED FOOD MKI67, FLOT1, VHL SIRT1 4382/4885KDM4E 3595/4885CYP1A2 2795/4885
US-12496357-B2 Compositions and methods for treating sickle cell disease HBB, HBG1, HBZ SIRT1 4760/4885KDM4E 4884/4885CYP1A2 4657/4885
US-20220378782-A1 KCC2 EXPRESSION ENHANCING COMPOUNDS AND USES THEREOF MECP2, SLC1A2, GRIN2C SIRT1 4028/4885KDM4E 127/4885CYP1A2 4732/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.