SCHEMBL25453063

SCHEMBL25453063

CN(c1cccc(Cl)c1)c1cc(N)ccn1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 3/20 0.46
GRM4 Q14833 1/20 0.45
GRM5 P41594 2/20 0.43
ALDH1A1 P00352 1/20 0.43
HTR3E A5X5Y0 1/20 0.43
HTR3B O95264 1/20 0.43
HTR3A P46098 1/20 0.43
HTR3D Q70Z44 1/20 0.43
HTR3C Q8WXA8 1/20 0.43
RXRA P19793 1/20 0.42
RXRB P28702 1/20 0.42
RXRG P48443 1/20 0.42
KDR P35968 3/20 0.42
FGFR1 P11362 1/20 0.42
EPHB4 P54760 1/20 0.42
CSF1R P07333 2/20 0.40
CHKA P35790 1/20 0.40
TAAR1 Q96RJ0 3/20 0.39
PDPK1 O15530 1/20 0.38
KIT P10721 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30502771 1.00 EGFR (0.46) EGFRGRM4GRM5ALDH1A1HTR3E
SCHEMBL25453062 0.83 KCNH2 (0.47) EGFRGRM5RXRAKDRCSF1R
SCHEMBL25453079 0.82 EGFR (0.48) EGFRALDH1A1RXRARXRBRXRG
SCHEMBL25175471 0.82 ALDH1A1 (0.47) EGFRGRM5ALDH1A1KDR
SCHEMBL26186425 0.79 P2RX4 (0.40) GRM4GRM5ALDH1A1HTR3EHTR3B
SCHEMBL4667357 0.77 ALDH1A1 (0.43) EGFRALDH1A1KDR
SCHEMBL4431783 0.77 KDR (0.50) EGFRGRM4GRM5HTR3EHTR3B
SCHEMBL25453064 0.73 GRIA1 (0.37) EGFRGRM5ALDH1A1
SCHEMBL7236726 0.73 CYP2D6 (0.41) EGFRALDH1A1KDRFGFR1
SCHEMBL2723906 0.71 PDPK1 (0.43) EGFRGRM4HTR3EHTR3BHTR3A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023081800-A1 ALPHA-2A ADRENERGIC RECEPTOR MODULATORS AND USES THEREOF THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2023-05-11 WO disclosed