SCHEMBL25453079

SCHEMBL25453079

CN(c1ccccc1)c1cc(N)ccn1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 2/20 0.48
ASIC3 Q9UHC3 2/20 0.46
DHFR P00374 3/20 0.42
CHKA P35790 1/20 0.41
OPRD1 P41143 1/20 0.39
ADORA2A P29274 1/20 0.38
ADORA1 P30542 1/20 0.38
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
FGFR1 P11362 1/20 0.36
KDR P35968 1/20 0.36
EPHB4 P54760 1/20 0.36
CYP1A2 P05177 2/20 0.36
CYP3A4 P08684 2/20 0.36
CYP2D6 P10635 2/20 0.36
CYP2C9 P11712 2/20 0.36
CYP2C19 P33261 2/20 0.36
L3MBTL1 Q9Y468 2/20 0.36
TSHR P16473 1/20 0.36
MAPK1 P28482 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4667357 0.87 ALDH1A1 (0.43) EGFRASIC3DHFRADORA2AADORA1
SCHEMBL25453062 0.83 KCNH2 (0.47) EGFRCHKAKDRTSHRMAPT
SCHEMBL25453064 0.83 GRIA1 (0.37) EGFRASIC3MEN1KMT2ACYP3A4
SCHEMBL30502771 0.82 EGFR (0.46) EGFRCHKAFGFR1KDREPHB4
SCHEMBL25175471 0.82 ALDH1A1 (0.47) EGFRASIC3OPRD1KDRCYP3A4
SCHEMBL25453063 0.82 EGFR (0.46) EGFRCHKAFGFR1KDREPHB4
SCHEMBL21241166 0.80 UHRF1 (0.42) EGFRDHFRCHKAMEN1KMT2A
SCHEMBL3658312 0.77 ADORA2A (0.44) ASIC3ADORA2AADORA1MEN1KMT2A
SCHEMBL7236726 0.76 CYP2D6 (0.41) EGFRDHFRMEN1KMT2AFGFR1
SCHEMBL26186404 0.76 OPRD1 (0.48) ASIC3OPRD1MEN1KMT2ATSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023081800-A1 ALPHA-2A ADRENERGIC RECEPTOR MODULATORS AND USES THEREOF THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2023-05-11 WO disclosed