SCHEMBL254610

SCHEMBL254610

C[C@@](O)(CF)[C@H](NC(=O)c1ccc(-c2ccc(N)cc2)cc1)C(=O)NO

nearest known ligand 0.52

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
ANPEP P15144 7/20 0.41
NPC1 O15118 1/20 0.40
RAB9A P51151 1/20 0.40
ESRRG P62508 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19262701 0.90
SCHEMBL159041 0.88
SCHEMBL15235779 0.88
SCHEMBL255220 0.86 NPC1 (0.41) NPC1RAB9AESRRG
SCHEMBL254947 0.85 NPC1 (0.40) NPC1RAB9AESRRG
SCHEMBL254900 0.84 ANPEP (0.39) ANPEPNPC1RAB9A
SCHEMBL13267172 0.83 NPC1 (0.41) ANPEPNPC1RAB9AESRRG
SCHEMBL255108 0.80 ANPEP (0.43) ANPEPNPC1RAB9AESRRG
SCHEMBL13459333 0.79 NPC1 (0.43) NPC1RAB9AESRRG
SCHEMBL19262877 0.78

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012031298-A2 ETHYNYLBENZENE DERIVATIVES DUKE UNIVERSITY (US) 2012-03-08 WO disclosed