SCHEMBL254947

SCHEMBL254947

COC(=O)[C@@H](NC(=O)c1ccc(-c2ccc(N)cc2)cc1)[C@](C)(O)CF

nearest known ligand 0.40

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.40
RAB9A P51151 2/20 0.40
ESRRG P62508 1/20 0.39
ADRB2 P07550 1/20 0.38
ADRB1 P08588 1/20 0.38
ADRB3 P13945 1/20 0.38
EPHX2 P34913 1/20 0.38
CYP26A1 O43174 1/20 0.37
CA2 P00918 1/20 0.36
MLYCD O95822 1/20 0.36
F10 P00742 4/20 0.36
PRSS1 P07477 3/20 0.36
F2 P00734 2/20 0.36
TSHR P16473 1/20 0.36
CYP3A4 P08684 2/20 0.35
LMNA P02545 1/20 0.35
CYP1A2 P05177 1/20 0.35
MAOA P21397 1/20 0.35
ALDH1A1 P00352 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15237910 0.88 ADRB2 (0.37) NPC1RAB9AESRRGADRB2ADRB1
SCHEMBL254376 0.86 CA2 (0.43) NPC1RAB9AESRRGADRB2ADRB1
SCHEMBL254610 0.85 ANPEP (0.41) NPC1RAB9AESRRG
SCHEMBL255310 0.84 NPC1 (0.38) NPC1RAB9AESRRGADRB2ADRB1
SCHEMBL254164 0.79 NPC1 (0.36) NPC1RAB9AESRRGADRB2ADRB1
SCHEMBL19262701 0.75
SCHEMBL159041 0.74
SCHEMBL15235779 0.74
SCHEMBL15235729 0.73 CA2 (0.39) NPC1RAB9AESRRGADRB2ADRB1
SCHEMBL255220 0.73 NPC1 (0.41) NPC1RAB9AESRRGCA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012031298-A2 ETHYNYLBENZENE DERIVATIVES DUKE UNIVERSITY (US) 2012-03-08 WO disclosed