SCHEMBL254640

SCHEMBL254640

COC(=O)[C@@H](NC(=O)c1ccc(C#Cc2ccc(N)cc2)cc1)C(C)(C)N

nearest known ligand 0.51

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ACACB O00763 1/20 0.41
ADRB2 P07550 1/20 0.40
ADRB1 P08588 1/20 0.40
ADRB3 P13945 1/20 0.40
APP P05067 1/20 0.39
NPC1 O15118 1/20 0.39
RAB9A P51151 1/20 0.39
RARB P10826 1/20 0.38
RARG P13631 1/20 0.38
CA2 P00918 1/20 0.38
ESRRG P62508 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20299901 1.00 ACACB (0.41) ACACBADRB2ADRB1ADRB3APP
SCHEMBL15235731 0.95 ADRB2 (0.38) ACACBADRB2ADRB1ADRB3NPC1
Trifluoroacetic Acid SCHEMBL20299911 0.93 NPC1 (0.39) ACACBNPC1RAB9ARARBRARG
SCHEMBL16840367 0.87 ACACB (0.38) ACACBRARBRARGCA2
SCHEMBL3017864 0.86 ACACB (0.46) ACACB
Hydrochloric Acid SCHEMBL16820709 0.86 ACACB (0.38) ACACBRARBRARGCA2
Hydrochloric Acid SCHEMBL16820710 0.86 ACACB (0.38) ACACBRARBRARGCA2
SCHEMBL15235729 0.85 CA2 (0.39) ACACBADRB2ADRB1ADRB3NPC1
SCHEMBL16840371 0.85 MMP2 (0.40) ACACBCA2
SCHEMBL20299876 0.85

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012031298-A2 ETHYNYLBENZENE DERIVATIVES DUKE UNIVERSITY (US) 2012-03-08 WO disclosed