SCHEMBL2547799

SCHEMBL2547799

COOC[Si](C)(C)c1ccccc1

nearest known ligand 0.39

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
MAPT P10636 1/20 0.39
ESR1 P03372 1/20 0.34
ESR2 Q92731 1/20 0.34
MGAM O43451 2/20 0.34
CA4 P22748 1/20 0.32
NR1H2 P55055 1/20 0.32
NR1H3 Q13133 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL40410 0.82 MAPT (0.41) MAPTESR1ESR2MGAMCA4
SCHEMBL40408 0.76 MAPT (0.40) MAPTESR1ESR2MGAMNR1H2
SCHEMBL11316383 0.74 MAPT (0.39) MAPTESR1ESR2MGAMNR1H2
SCHEMBL869282 0.74 MAPT (0.39) MAPTESR1ESR2MGAMNR1H2
SCHEMBL2355439 0.72 MAPT (0.42) MAPTESR1ESR2MGAMNR1H2
SCHEMBL1470884 0.72 MAPT (0.38) MAPTESR1ESR2MGAMNR1H2
SCHEMBL16325251 0.72 MAPT (0.38) MAPTESR1ESR2MGAMNR1H2
SCHEMBL7033371 0.72 MAPT (0.42) MAPTESR1ESR2MGAMNR1H2
SCHEMBL11316112 0.71 MAPT (0.41) MAPTESR1ESR2MGAMNR1H2
SCHEMBL9217667 0.71 MAPT (0.47) MAPTESR1ESR2MGAMNR1H2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111330016-A Antibody Drug Conjugates (ADC) that bind to 158P1D7 protein 艾更斯司股份有限公司 2020-06-26 CN disclosed
CN-111330017-A Antibody Drug Conjugates (ADC) that bind to 158P1D7 protein 艾更斯司股份有限公司 2020-06-26 CN disclosed
CN-105073132-B Antibody Drug Conjugates (ADC) that bind to 158P1D7 protein 艾更斯司股份有限公司 2020-01-10 CN disclosed
EP-2560634-A1 NITRIC OXIDE RELEASING PRODRUGS OF THERAPEUTIC AGENTS Piramal Enterprises Limited (IN) 2013-02-27 EP disclosed
WO-2011132171-A1 NITRIC OXIDE RELEASING PRODRUGS OF THERAPEUTIC AGENTS PIRAMAL LIFE SCIENCES LIMITED (IN) 2011-10-27 WO disclosed
US-20110263526-A1 Nitric Oxide Releasing Prodrugs of Therapeutic Agents PIRAMAL LIFE SCIENCES LIMITED (IN) 2011-10-27 US disclosed
EP-1896480-A1 CRIPOWELLINS AND SYNTHETIC DERIVATIVES THEREOF USED AS MEDICAMENTS Bayer CropScience Aktiengesellschaft (DE) 2008-03-12 EP disclosed
WO-2006136309-A1 CRIPOWELLINS AND SYNTHETIC DERIVATIVES THEREOF USED AS MEDICAMENTS BAYER CROPSCIENCE AKTIENGESELLSCHAFT (DE) 2006-12-28 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110263526-A1 Nitric Oxide Releasing Prodrugs of Therapeutic Agents NOS2, NOS1, NOS3 MAPT 4304/4885ESR1 1694/4885ESR2 1855/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.