SCHEMBL2549332

SCHEMBL2549332

ClC1(c2ccc3c(c2)CN(c2ccccn2)Cc2nncn2-3)CCC(c2ccccc2)CC1

nearest known ligand 0.38

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
AVPR1A P37288 13/20 0.37
AVPR2 P30518 9/20 0.37
KCNH2 Q12809 4/20 0.37
OXTR P30559 3/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL2551680 0.78 OPRK1 (0.34) AVPR1A
SCHEMBL2552411 0.75 AVPR1A (0.34) AVPR1AKCNH2
SCHEMBL2567189 0.75 AVPR1A (0.38) AVPR1A
Hydrochloric Acid SCHEMBL2563942 0.74 AVPR1A (0.37) AVPR1A
SCHEMBL2564920 0.73 AVPR1A (0.35) AVPR1A
SCHEMBL2556524 0.72 CYP11B2 (0.32) AVPR1AAVPR2KCNH2
SCHEMBL2565904 0.72 AVPR2 (0.37) AVPR1AAVPR2KCNH2OXTR
SCHEMBL2590577 0.71 AVPR1A (0.32) AVPR1AAVPR2KCNH2
SCHEMBL2563262 0.71 CYP11B2 (0.41) AVPR1A
SCHEMBL2579657 0.71 OXTR (0.36) AVPR1AAVPR2KCNH2OXTR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2552919-A1 ARYL-CYCLOHEXYL-TETRAAZABENZO[E]AZULENES F. Hoffmann-La Roche AG (CH) 2013-02-06 EP disclosed
WO-2011120877-A1 ARYL-CYCLOHEXYL-TETRAAZABENZO[E]AZULENES F. HOFFMANN-LA ROCHE AG (CH) 2011-10-06 WO disclosed