SCHEMBL25516110

SCHEMBL25516110

CC(=N)c1cc(C(N)=O)ccc1N

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.41
ALDH1A1 P00352 2/20 0.41
HSD17B10 Q99714 2/20 0.41
PARP1 P09874 4/20 0.40
IKBKB O14920 1/20 0.40
MAPT P10636 3/20 0.39
NPC1 O15118 1/20 0.39
MAPK1 P28482 1/20 0.39
HTT P42858 1/20 0.39
NOS1 P29475 1/20 0.39
LCK P06239 1/20 0.39
BRD4 O60885 1/20 0.39
BRPF1 P55201 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
F2 P00734 1/20 0.38
PRSS1 P07477 1/20 0.38
PRSS2 P07478 1/20 0.38
PRSS3 P35030 1/20 0.38
ST14 Q9Y5Y6 1/20 0.38
KMT2A Q03164 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13522728 0.85 CDC25B (0.49) KDM4EALDH1A1HSD17B10MAPTNPC1
SCHEMBL1805758 0.82 IKBKB (0.55) KDM4EALDH1A1HSD17B10PARP1IKBKB
SCHEMBL24633560 0.81 ALDH1A1 (0.44) KDM4EALDH1A1MAPTNPC1MAPK1
SCHEMBL22489533 0.81 ALDH1A1 (0.60) KDM4EALDH1A1HSD17B10MAPTNPC1
SCHEMBL25516265 0.81 MAPT (0.43) KDM4EALDH1A1HSD17B10MAPTHTT
SCHEMBL25515246 0.75 MAPT (0.34) KDM4EALDH1A1HSD17B10MAPTNPC1
SCHEMBL12073780 0.75 CHEK2 (0.40) KDM4E
SCHEMBL27448425 0.74 ALDH1A1 (0.41) KDM4EALDH1A1HSD17B10PARP1IKBKB
SCHEMBL22890834 0.74 THRB (0.52) KDM4EALDH1A1HSD17B10MAPTF2
SCHEMBL8412857 0.73 ALDH1A1 (0.49) KDM4EALDH1A1HSD17B10PARP1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023078337-A1 CDK8/19 DUAL INHIBITORS AND METHODS OF USE INSILICO MEDICINE IP LIMITED (CN) 2023-05-11 WO disclosed