SCHEMBL25523929

SCHEMBL25523929

COc1ccn2c([C@H]3CCC[C@@H](N)C3)nnc2c1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRM2 Q14416 1/20 0.40
MAPK13 O15264 3/20 0.37
ADORA2A P29274 4/20 0.36
ALDH1A1 P00352 2/20 0.35
HPGD P15428 2/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
LRRK2 Q5S007 1/20 0.34
TNK2 Q07912 2/20 0.34
NOS3 P29474 2/20 0.34
NOS1 P29475 2/20 0.34
NOS2 P35228 2/20 0.34
ADORA3 P0DMS8 1/20 0.33
MAPT P10636 2/20 0.33
POLB P06746 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
PDE10A Q9Y233 1/20 0.33
CCNT1 O60563 1/20 0.33
CDK9 P50750 1/20 0.33
AKT1 P31749 1/20 0.33
AKT2 P31751 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25533147 0.85 GRM2 (0.38) GRM2MAPK13
SCHEMBL25526353 0.81 GRM2 (0.43) GRM2MAPK13
SCHEMBL30397943 0.80 MAPK13 (0.41) GRM2MAPK13ADORA2A
SCHEMBL30397669 0.80 MAPK13 (0.41) GRM2MAPK13ADORA2A
SCHEMBL25522679 0.78 GRM2 (0.40) GRM2MAPK13LRRK2TNK2NOS3
SCHEMBL25521381 0.78 GRM2 (0.40) GRM2MAPK13LRRK2TNK2NOS3
SCHEMBL30397855 0.77 MAPK14 (0.42) GRM2ALDH1A1HPGDSMN1; SMN2
SCHEMBL25516112 0.77 MAPK14 (0.42) GRM2ALDH1A1HPGDSMN1; SMN2
SCHEMBL25532532 0.77 MAPK14 (0.42) GRM2ALDH1A1HPGDSMN1; SMN2
SCHEMBL30397394 0.76 GRM2 (0.37) GRM2MAPK13ADORA2AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023091726-A1 INHIBITORS OF CYCLIN‑DEPENDENT KINASE 12 (CDK12) SYROS PHARMACEUTICALS, INC. (US) 2023-05-25 WO disclosed