SCHEMBL25528332

SCHEMBL25528332

C[C@H](CO)NC(=O)c1cccc(CN2C(=O)c3ccc(-c4ccnc(N)c4)cc3N(C)C(=O)[C@H]2C)c1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 7/20 0.38
ROCK1 Q13464 5/20 0.38
CYP3A4 P08684 1/20 0.37
CYP2D6 P10635 1/20 0.37
MAP4K4 O95819 1/20 0.36
ALOX5AP P20292 3/20 0.34
FEN1 P39748 3/20 0.34
MAPK3 P27361 1/20 0.34
MAPK1 P28482 1/20 0.34
CIT O14578 1/20 0.33
AGTR2 P50052 1/20 0.33
PRKAG1 P54619 1/20 0.33
PRKAA2 P54646 1/20 0.33
PRKAB1 Q9Y478 1/20 0.33
LARS1 Q9P2J5 1/20 0.33
SYK P43405 1/20 0.33
REN P00797 2/20 0.33
ADORA3 P0DMS8 1/20 0.33
ADORA2A P29274 1/20 0.33
ADORA2B P29275 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25528328 0.88 BRD4 (0.43) ROCK2ROCK1CYP3A4
SCHEMBL25528623 0.86 ROCK2 (0.35) ROCK2ROCK1CYP3A4CYP2D6AGTR2
SCHEMBL25528333 0.86 ROCK2 (0.39) ROCK2ROCK1
SCHEMBL25528200 0.85 ROCK2 (0.40) ROCK2ROCK1MAP4K4
SCHEMBL25528201 0.84 ROCK2 (0.39) ROCK2ROCK1MAP4K4
SCHEMBL25528196 0.83 ROCK2 (0.43) ROCK2ROCK1MAP4K4
SCHEMBL25529691 0.82 ROCK2 (0.40) ROCK2ROCK1
SCHEMBL25528334 0.81 NPSR1 (0.45) ROCK2ROCK1MAP4K4ADORA2AADORA1
SCHEMBL25528181 0.79 ROCK2 (0.59) ROCK2ROCK1CYP3A4
SCHEMBL25528180 0.79 ROCK2 (0.59) ROCK2ROCK1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023093787-A1 BENZODIAZEPINE COMPOUND AND APPLICATION THEREOF AS RHO KINASE INHIBITOR 成都奥睿药业有限公司 2023-06-01 WO disclosed