SCHEMBL25528334

SCHEMBL25528334

C[C@@H]1C(=O)N(C)c2cc(-c3ccnc(N)c3)ccc2C(=O)N1Cc1cccc(C(=O)NCCN2CCOCC2)c1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 1/20 0.45
HPGDS O60760 2/20 0.43
CYP2C9 P11712 1/20 0.42
CYP2C19 P33261 1/20 0.42
ERN1 O75460 1/20 0.42
ROCK2 O75116 1/20 0.42
ROCK1 Q13464 1/20 0.42
MAP4K4 O95819 1/20 0.42
ALDH1A1 P00352 2/20 0.42
PARP1 P09874 1/20 0.41
ADORA2A P29274 1/20 0.41
ADORA1 P30542 1/20 0.41
LMNA P02545 1/20 0.41
TP53 P04637 1/20 0.41
KMT2A Q03164 1/20 0.41
HTT P42858 1/20 0.41
CD274 Q9NZQ7 2/20 0.41
CACNA1G O43497 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
GRK5 P34947 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25529165 0.91 NPSR1 (0.44) NPSR1HPGDSCYP2C9CYP2C19ERN1
SCHEMBL25528328 0.87 BRD4 (0.43) ROCK2ROCK1
SCHEMBL25528200 0.86 ROCK2 (0.40) ROCK2ROCK1MAP4K4PARP1KMT2A
SCHEMBL25528333 0.85 ROCK2 (0.39) ROCK2ROCK1
SCHEMBL25528196 0.85 ROCK2 (0.43) ROCK2ROCK1MAP4K4PARP1
SCHEMBL25528201 0.84 ROCK2 (0.39) ROCK2ROCK1MAP4K4PARP1KMT2A
SCHEMBL25528332 0.81 ROCK2 (0.38) ROCK2ROCK1MAP4K4ADORA2AADORA1
SCHEMBL25529691 0.79 ROCK2 (0.40) ROCK2ROCK1
SCHEMBL25528181 0.76 ROCK2 (0.59) ROCK2ROCK1
SCHEMBL25528180 0.76 ROCK2 (0.59) ROCK2ROCK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023093787-A1 BENZODIAZEPINE COMPOUND AND APPLICATION THEREOF AS RHO KINASE INHIBITOR 成都奥睿药业有限公司 2023-06-01 WO disclosed