SCHEMBL25528344

SCHEMBL25528344

CN/C(=C\C=N)c1ccc2c(c1)N(C)C(=O)[C@@H](C)N(Cc1cc(F)cc(C(=O)NCC3CCN(C)CC3)c1)C2=O

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAP4K4 O95819 1/20 0.36
PARP1 P09874 1/20 0.34
CACNA1H O95180 2/20 0.33
CDK1 P06493 1/20 0.33
CCNB1 P14635 1/20 0.33
CCNA2 P20248 1/20 0.33
CDK2 P24941 1/20 0.33
PDGFRB P09619 1/20 0.33
FGFR1 P11362 1/20 0.33
KDR P35968 1/20 0.33
BRD4 O60885 3/20 0.33
CACNA1G O43497 3/20 0.33
CACNA1I Q9P0X4 2/20 0.33
NAMPT P43490 2/20 0.33
HDAC4 P56524 1/20 0.33
LMNA P02545 1/20 0.32
GAA P10253 1/20 0.32
KCNH2 Q12809 1/20 0.32
EGLN1 Q9GZT9 1/20 0.31
USP30 Q70CQ3 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25528752 0.90 PARP1 (0.42) MAP4K4PARP1BRD4CACNA1GCACNA1I
SCHEMBL25528767 0.88 MAP4K4 (0.38) MAP4K4PARP1CACNA1HCDK1CCNB1
SCHEMBL25529759 0.80 MAP4K4 (0.40) MAP4K4PARP1CACNA1HCDK1CCNB1
SCHEMBL25528758 0.79 PARP1 (0.42) MAP4K4PARP1BRD4CACNA1GNAMPT
SCHEMBL25528339 0.77 PARP1 (0.41) MAP4K4PARP1BRD4CACNA1GNAMPT
SCHEMBL25528470 0.75 AURKA (0.37) MAP4K4CACNA1HEGLN1USP30ROCK2
SCHEMBL25528475 0.72 CACNA1H (0.36) MAP4K4CACNA1HUSP30ROCK2
SCHEMBL25531283 0.72 CACNA1H (0.36) MAP4K4CACNA1HUSP30ROCK2
SCHEMBL25532516 0.72 ROCK2 (0.43) PARP1BRD4CACNA1INAMPTHDAC4
SCHEMBL25528762 0.72 CACNA1H (0.34) MAP4K4CACNA1HCDK1CCNB1CCNA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023093787-A1 BENZODIAZEPINE COMPOUND AND APPLICATION THEREOF AS RHO KINASE INHIBITOR 成都奥睿药业有限公司 2023-06-01 WO disclosed