SCHEMBL25529759

SCHEMBL25529759

C[C@@H]1C(=O)N(C)c2cc(-c3ccnn3C)ccc2C(=O)N1Cc1cc(F)cc(C(=O)NCC2CCN(C)CC2)c1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAP4K4 O95819 1/20 0.40
HDAC4 P56524 1/20 0.38
ROCK2 O75116 3/20 0.36
CDK1 P06493 1/20 0.36
CCNB1 P14635 1/20 0.36
CCNA2 P20248 1/20 0.36
CDK2 P24941 1/20 0.36
BRD4 O60885 1/20 0.35
EGLN1 Q9GZT9 3/20 0.35
PARP1 P09874 1/20 0.34
CD274 Q9NZQ7 1/20 0.34
CACNA1H O95180 2/20 0.33
AKT1 P31749 2/20 0.33
AKT2 P31751 2/20 0.33
WDR5 P61964 1/20 0.33
KMT2A Q03164 1/20 0.33
GSK3B P49841 1/20 0.33
DYRK1A Q13627 1/20 0.33
CACNA1G O43497 1/20 0.33
CACNA1I Q9P0X4 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25528771 0.86 ROCK2 (0.42) HDAC4ROCK2BRD4PARP1
SCHEMBL25528470 0.82 AURKA (0.37) MAP4K4ROCK2EGLN1CACNA1H
SCHEMBL25528762 0.81 CACNA1H (0.34) MAP4K4CDK1CCNB1CCNA2CDK2
SCHEMBL25531283 0.80 CACNA1H (0.36) MAP4K4ROCK2CACNA1H
SCHEMBL25528475 0.80 CACNA1H (0.36) MAP4K4ROCK2CACNA1H
SCHEMBL25528344 0.80 MAP4K4 (0.36) MAP4K4HDAC4ROCK2CDK1CCNB1
SCHEMBL25532516 0.80 ROCK2 (0.43) HDAC4ROCK2BRD4EGLN1PARP1
SCHEMBL25528767 0.80 MAP4K4 (0.38) MAP4K4HDAC4CDK1CCNB1CCNA2
SCHEMBL25528468 0.79 CACNA1H (0.36) CACNA1HWDR5
SCHEMBL25528343 0.78 PARP1 (0.43) MAP4K4HDAC4ROCK2CDK1CCNB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023093787-A1 BENZODIAZEPINE COMPOUND AND APPLICATION THEREOF AS RHO KINASE INHIBITOR 成都奥睿药业有限公司 2023-06-01 WO disclosed