SCHEMBL25528762

SCHEMBL25528762

Cc1cnn(C)c1-c1ccc2c(c1)N(C)C(=O)[C@@H](C)N(Cc1cc(F)cc(C(=O)NCC3CCN(C)C(C)C3)c1)C2=O

nearest known ligand 0.34

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CACNA1H O95180 4/20 0.34
LMNA P02545 1/20 0.34
GAA P10253 1/20 0.34
MAP4K4 O95819 1/20 0.32
CTSC P53634 1/20 0.32
CDK1 P06493 1/20 0.31
CCNB1 P14635 1/20 0.31
CCNA2 P20248 1/20 0.31
CDK2 P24941 1/20 0.31
USP30 Q70CQ3 1/20 0.31
KCNH2 Q12809 1/20 0.30
CACNA1I Q9P0X4 1/20 0.30
EGLN1 Q9GZT9 2/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25528468 0.91 CACNA1H (0.36) CACNA1HLMNAGAACTSC
SCHEMBL25528830 0.84 HPGD (0.33)
SCHEMBL25528465 0.84 CACNA1H (0.33) CACNA1H
SCHEMBL25528343 0.83 PARP1 (0.43) MAP4K4CDK1CCNB1CCNA2CDK2
SCHEMBL25528466 0.81 ROCK2 (0.37) CACNA1HGAA
SCHEMBL25529759 0.81 MAP4K4 (0.40) CACNA1HMAP4K4CDK1CCNB1CCNA2
SCHEMBL25528467 0.78 HTR7 (0.34)
SCHEMBL25528475 0.77 CACNA1H (0.36) CACNA1HMAP4K4USP30
SCHEMBL25531283 0.77 CACNA1H (0.36) CACNA1HMAP4K4USP30
SCHEMBL25528470 0.77 AURKA (0.37) CACNA1HMAP4K4USP30EGLN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023093787-A1 BENZODIAZEPINE COMPOUND AND APPLICATION THEREOF AS RHO KINASE INHIBITOR 成都奥睿药业有限公司 2023-06-01 WO disclosed