SCHEMBL25528834

SCHEMBL25528834

Cc1ccc(C(=O)OC(C)CNC(=O)c2cccc(CN3C(=O)c4ccc(-c5c(C)cnn5C)cc4N(C)C(=O)[C@H]3C)c2)c(C)c1

nearest known ligand 0.33

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
HTR7 P34969 1/20 0.33
POLB P06746 1/20 0.33
CACNA1G O43497 4/20 0.32
BRD4 O60885 2/20 0.32
THRB P10828 1/20 0.31
PRKAG1 P54619 1/20 0.31
PRKAA2 P54646 1/20 0.31
PRKAB1 Q9Y478 1/20 0.31
ROCK2 O75116 5/20 0.31
ROCK1 Q13464 5/20 0.31
GAA P10253 1/20 0.31
LMNA P02545 1/20 0.31
KDM4E B2RXH2 1/20 0.31
ALDH1A1 P00352 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25528467 0.91 HTR7 (0.34) HTR7
SCHEMBL25528469 0.87 POLB (0.36) POLBCACNA1GBRD4THRBROCK2
SCHEMBL25528346 0.86 ROCK2 (0.36) CACNA1GBRD4THRBROCK2ROCK1
SCHEMBL25528831 0.81 HTR7 (0.36) HTR7BRD4ROCK2ROCK1
SCHEMBL25528466 0.80 ROCK2 (0.37) CACNA1GBRD4THRBROCK2ROCK1
SCHEMBL25529880 0.79 HTR7 (0.33) HTR7
SCHEMBL25528343 0.79 PARP1 (0.43) BRD4ROCK2ROCK1
SCHEMBL25528465 0.78 CACNA1H (0.33) BRD4
SCHEMBL25528830 0.78 HPGD (0.33)
SCHEMBL25528478 0.76 ROCK2 (0.41) CACNA1GBRD4THRBROCK2ROCK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023093787-A1 BENZODIAZEPINE COMPOUND AND APPLICATION THEREOF AS RHO KINASE INHIBITOR 成都奥睿药业有限公司 2023-06-01 WO disclosed