SCHEMBL25528469

SCHEMBL25528469

Cc1cnn(C)c1-c1ccc2c(c1)N(C)C(=O)[C@@H](C)N(Cc1cccc(C(=O)NCC(C)O)c1)C2=O

nearest known ligand 0.36

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
POLB P06746 1/20 0.36
LMNA P02545 1/20 0.36
HPGD P15428 1/20 0.35
ALDH1A1 P00352 1/20 0.33
KDM4E B2RXH2 1/20 0.32
CACNA1G O43497 4/20 0.32
BRD4 O60885 3/20 0.32
WNT1 P04628 1/20 0.32
CLK2 P49760 1/20 0.32
CLK3 P49761 1/20 0.32
GSK3B P49841 1/20 0.32
DYRK1A Q13627 1/20 0.32
IRAK4 Q9NWZ3 1/20 0.32
ROCK2 O75116 3/20 0.32
ROCK1 Q13464 3/20 0.32
PRMT5 O14744 1/20 0.32
MAPK14 Q16539 1/20 0.32
THRB P10828 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25528830 0.90 HPGD (0.33) HPGD
SCHEMBL25528834 0.87 HTR7 (0.33) POLBLMNAALDH1A1KDM4ECACNA1G
SCHEMBL25528466 0.86 ROCK2 (0.37) ALDH1A1CACNA1GBRD4WNT1CLK2
SCHEMBL25528343 0.86 PARP1 (0.43) BRD4GSK3BROCK2ROCK1MAPK14
SCHEMBL25528346 0.80 ROCK2 (0.36) KDM4ECACNA1GBRD4ROCK2ROCK1
SCHEMBL25528467 0.78 HTR7 (0.34)
SCHEMBL25528468 0.77 CACNA1H (0.36) LMNAMAPK14
SCHEMBL25529692 0.75 ROCK2 (0.52) ROCK2ROCK1
SCHEMBL25528771 0.75 ROCK2 (0.42) BRD4ROCK2ROCK1MAPK14
SCHEMBL25528328 0.73 BRD4 (0.43) BRD4ROCK2ROCK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023093787-A1 BENZODIAZEPINE COMPOUND AND APPLICATION THEREOF AS RHO KINASE INHIBITOR 成都奥睿药业有限公司 2023-06-01 WO disclosed