SCHEMBL25528835

SCHEMBL25528835

Cc1ccc(C(=O)OCC(C)(C)CNC(=O)c2cc(F)cc(CN3C(=O)c4ccc(-c5ccncc5)cc4N(C)C(=O)[C@H]3C)c2)c(C)c1

nearest known ligand 0.32

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 1/20 0.32
ROCK1 Q13464 1/20 0.32
AURKA O14965 1/20 0.30
BRD4 O60885 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25528611 0.88 ROCK1 (0.33) ROCK2ROCK1AURKA
SCHEMBL25528837 0.87 ROCK2 (0.32) ROCK2ROCK1BRD4
SCHEMBL25528831 0.86 HTR7 (0.36) ROCK2ROCK1AURKABRD4
SCHEMBL25529070 0.85 CACNA1H (0.33) ROCK2ROCK1AURKABRD4
SCHEMBL25528479 0.85 CACNA1H (0.33) ROCK2ROCK1AURKABRD4
SCHEMBL25528845 0.84 ROCK2 (0.32) ROCK2ROCK1AURKA
SCHEMBL25528839 0.84 F10 (0.34) ROCK2ROCK1BRD4
SCHEMBL25528750 0.81 ROCK2 (0.33) ROCK2ROCK1BRD4
SCHEMBL25528842 0.79 ROCK2 (0.41) ROCK2ROCK1AURKA
SCHEMBL25528475 0.77 CACNA1H (0.36) ROCK2ROCK1AURKA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023093787-A1 BENZODIAZEPINE COMPOUND AND APPLICATION THEREOF AS RHO KINASE INHIBITOR 成都奥睿药业有限公司 2023-06-01 WO disclosed