SCHEMBL25530648

SCHEMBL25530648

COC(=O)c1cccc(CN2C(=O)c3ccc(Br)cc3N(C)C(=O)[C@H]2CO)c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 6/20 0.47
MAPK8 P45983 1/20 0.43
TRPA1 O75762 1/20 0.42
CYP4F2 P78329 2/20 0.41
CYP4A11 Q02928 2/20 0.41
L3MBTL1 Q9Y468 1/20 0.40
MAPK10 P53779 1/20 0.40
BACE1 P56817 2/20 0.40
POLB P06746 2/20 0.39
ROCK2 O75116 1/20 0.39
ROCK1 Q13464 1/20 0.39
GAA P10253 1/20 0.39
ABHD6 Q9BV23 1/20 0.39
LOXL2 Q9Y4K0 1/20 0.39
IDO1 P14902 1/20 0.39
THRB P10828 1/20 0.39
GSK3B P49841 1/20 0.38
CD74 P04233 1/20 0.38
MIF P14174 1/20 0.38
CASP3 P42574 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25529498 0.89 MAPT (0.48) MAPTMAPK8TRPA1CYP4F2CYP4A11
SCHEMBL25530633 0.82 ROCK2 (0.45) MAPTTRPA1CYP4F2CYP4A11L3MBTL1
SCHEMBL25529500 0.74 ROCK2 (0.59) MAPTTRPA1L3MBTL1MAPK10POLB
SCHEMBL25530634 0.72 ROCK2 (0.40) ROCK2ROCK1IDO1
SCHEMBL25530880 0.71 ROCK1 (0.48) MAPTTRPA1L3MBTL1MAPK10POLB
SCHEMBL28799626 0.71 ALDH1A1 (0.62) MAPTMAPK8TRPA1L3MBTL1IDO1
SCHEMBL15523614 0.67 MAPT (0.53) MAPTMAPK8CYP4F2CYP4A11MAPK10
SCHEMBL31753576 0.66 KMT2A (0.70) MAPTTRPA1CYP4F2CYP4A11L3MBTL1
SCHEMBL1164954 0.66 KMT2A (0.70) MAPTTRPA1CYP4F2CYP4A11L3MBTL1
SCHEMBL6179524 0.64 MAPK8 (0.56) MAPTMAPK8CYP4F2CYP4A11MAPK10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023093787-A1 BENZODIAZEPINE COMPOUND AND APPLICATION THEREOF AS RHO KINASE INHIBITOR 成都奥睿药业有限公司 2023-06-01 WO disclosed