SCHEMBL25530633

SCHEMBL25530633

COC(=O)c1cccc(CN2C(=O)c3ccc(-c4ccnc(N)c4)cc3N(C)C(=O)[C@H]2CO)c1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 8/20 0.45
ROCK1 Q13464 4/20 0.45
TNIK Q9UKE5 1/20 0.39
CD74 P04233 1/20 0.39
MIF P14174 1/20 0.39
TRPA1 O75762 1/20 0.39
IDO1 P14902 1/20 0.38
KDM4E B2RXH2 1/20 0.37
GAA P10253 1/20 0.37
CASP7 P55210 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37
MAPK10 P53779 1/20 0.37
ABHD6 Q9BV23 1/20 0.36
CYP3A4 P08684 1/20 0.36
PRKACA P17612 1/20 0.36
LOXL2 Q9Y4K0 1/20 0.36
MAPT P10636 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
CYP4F2 P78329 1/20 0.35
CYP4A11 Q02928 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25530634 0.91 ROCK2 (0.40) ROCK2ROCK1IDO1
SCHEMBL25530636 0.84 ROCK2 (0.43) ROCK2ROCK1
SCHEMBL25530648 0.82 MAPT (0.47) ROCK2ROCK1CD74MIFTRPA1
SCHEMBL25530880 0.81 ROCK1 (0.48) ROCK2ROCK1TNIKCD74MIF
SCHEMBL25528651 0.80 ROCK2 (0.38) ROCK2ROCK1
SCHEMBL25529500 0.80 ROCK2 (0.59) ROCK2ROCK1TNIKCD74MIF
SCHEMBL25528328 0.79 BRD4 (0.43) ROCK2ROCK1CYP3A4
SCHEMBL25530811 0.79 BRD4 (0.49) ROCK2ROCK1MAPK10
SCHEMBL25528332 0.79 ROCK2 (0.38) ROCK2ROCK1CYP3A4ADORA2AADORA1
SCHEMBL25528181 0.77 ROCK2 (0.59) ROCK2ROCK1TNIKCYP3A4PRKACA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023093787-A1 BENZODIAZEPINE COMPOUND AND APPLICATION THEREOF AS RHO KINASE INHIBITOR 成都奥睿药业有限公司 2023-06-01 WO disclosed