SCHEMBL25533792

SCHEMBL25533792

CC(=O)N1C[C@@H](Nc2ncc(C(F)(F)F)cn2)C[C@@H](c2nnc3cc(C#N)ccn23)C1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IGF1R P08069 1/20 0.36
HCRTR1 O43613 3/20 0.35
MAP3K12 Q12852 2/20 0.34
EGLN2 Q96KS0 1/20 0.34
IRAK4 Q9NWZ3 2/20 0.33
CCNK O75909 5/20 0.33
CDK12 Q9NYV4 5/20 0.33
BRD4 O60885 1/20 0.33
CHRM2 P08172 1/20 0.33
CHRM1 P11229 1/20 0.33
CHRM3 P20309 1/20 0.33
CDK7 P50613 2/20 0.33
CCNH P51946 2/20 0.33
MNAT1 P51948 2/20 0.33
CCNT1 O60563 1/20 0.33
CCNE1 P24864 1/20 0.33
CDK2 P24941 1/20 0.33
CDK9 P50750 1/20 0.33
KCNJ5 P48544 1/20 0.33
MAPK3 P27361 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30398131 0.92 CHRM2 (0.35) IGF1RHCRTR1CCNKCDK12CHRM2
SCHEMBL25533466 0.90 GPR119 (0.38) HCRTR1EGLN2IRAK4
SCHEMBL25417681 0.81 CCNK (0.48) CCNKCDK12CDK7CCNHMNAT1
SCHEMBL30397353 0.75 CCR6 (0.44) HCRTR1CCR6
SCHEMBL30397120 0.70 CDK7 (0.36) CCNKCDK12CDK7CCNHMNAT1
SCHEMBL30397946 0.69 CDK7 (0.38) CCNKCDK12CDK7CCNHMNAT1
SCHEMBL30397422 0.68 CCNK (0.34) HCRTR1CCNKCDK12CDK7CCNH
SCHEMBL30396777 0.68 CCNK (0.39) CCNKCDK12CDK7CCNHMNAT1
SCHEMBL25517516 0.67 DRD2 (0.43) IRAK4F2R
SCHEMBL30397242 0.67 DPP4 (0.38) HCRTR1CCR6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023091726-A1 INHIBITORS OF CYCLIN‑DEPENDENT KINASE 12 (CDK12) SYROS PHARMACEUTICALS, INC. (US) 2023-05-25 WO disclosed