SCHEMBL255485

SCHEMBL255485

CC(C)(C)OC(=O)N1CCN(c2ccc(N)nc2)C(=O)C1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 2/20 0.44
NR1H2 P55055 2/20 0.44
ALDH1A1 P00352 1/20 0.44
LMNA P02545 1/20 0.44
MEN1 O00255 1/20 0.41
TSHR P16473 1/20 0.41
KMT2A Q03164 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
GPR119 Q8TDV5 4/20 0.41
MAP4K4 O95819 1/20 0.40
ENPP2 Q13822 2/20 0.40
HRH3 Q9Y5N1 1/20 0.40
POLB P06746 1/20 0.40
PTPN11 Q06124 1/20 0.39
CKS1B P61024 1/20 0.39
SKP1 P63208 1/20 0.39
SKP2 Q13309 1/20 0.39
ESR2 Q92731 1/20 0.39
PIK3CA P42336 1/20 0.39
ADORA1 P30542 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29491152 1.00 MAPT (0.44) MAPTNR1H2ALDH1A1LMNAMEN1
SCHEMBL18291495 0.93 NR1H2 (0.42) MAPTNR1H2ALDH1A1LMNAMEN1
SCHEMBL20037632 0.89 MAPT (0.43) MAPTNR1H2ALDH1A1LMNAMEN1
SCHEMBL14845641 0.88 MAPT (0.48) MAPTNR1H2ALDH1A1LMNAMEN1
SCHEMBL22650785 0.87 POLB (0.44) MAPTNR1H2ALDH1A1LMNAMEN1
SCHEMBL29462384 0.87 POLB (0.44) MAPTNR1H2ALDH1A1LMNAMEN1
SCHEMBL1584044 0.86 GPR119 (0.48) MAPTNR1H2ALDH1A1LMNAMEN1
SCHEMBL255156 0.84 MAPT (0.51) MAPTNR1H2ALDH1A1LMNAMEN1
SCHEMBL29491170 0.84 MAPT (0.51) MAPTNR1H2ALDH1A1LMNAMEN1
SCHEMBL76458 0.84 NR1H2 (0.54) MAPTNR1H2ALDH1A1LMNAGPR119

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 98 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20260146042-A1 PYRROLOPYRIMIDINE COMPOUNDS AND THEIR USES NOVARTIS AG (CH) 2026-05-28 US disclosed
WO-2025235363-A1 CYCLIN-DEPENDENT KINASE 4 DEGRADERS BLUEPRINT MEDICINES CORPORATION (US) 2025-11-13 WO disclosed
CN-120040446-A CDK inhibitors 基因泰克公司 2025-05-27 CN disclosed
US-20240043428-A1 PYRROLOPYRIMIDINE COMPOUNDS AND THEIR USES ASTEX THERAPEUTICS LTD. (GB) 2024-02-08 US disclosed
US-20230062022-A1 HETEROCYCLIC COMPOUNDS AS KINASE INHIBITORS NUVATION BIO INC (US) 2023-03-02 US disclosed
US-20230062022-A1 HETEROCYCLIC COMPOUNDS AS KINASE INHIBITORS NUVATION BIO INC (US) 2023-03-02 US disclosed
US-20220296595-A1 CDK INHIBITORS GENENTECH, INC. 2022-09-22 US disclosed
CN-110036012-B Pyrido [3,4-d ] pyrimidine derivatives and pharmaceutically acceptable salts thereof 帝人制药株式会社 2022-05-10 CN disclosed
CN-114364675-A CDK inhibitors 上海齐鲁锐格医药研发有限公司 2022-04-15 CN disclosed
US-11261182-B2 Crystal of pyrido[3,4-d]pyrimidine derivative or solvate thereof TEIJIN PHARMA LIMITED (JP) 2022-03-01 US disclosed
US-20110152244-A1 PYRROLOPYRIMIDINE COMPOUNDS AND THEIR USES NOVARTIS AG (CH) 2011-06-23 US disclosed
US-20110152244-A1 PYRROLOPYRIMIDINE COMPOUNDS AND THEIR USES NOVARTIS AG (CH) 2011-06-23 US disclosed
US-20110152244-A1 PYRROLOPYRIMIDINE COMPOUNDS AND THEIR USES NOVARTIS AG (CH) 2011-06-23 US disclosed
EP-2331547-A1 PYRROLOPYRIMIDINE COMPOUNDS AS CDK INHIBITORS Novartis AG (CH) 2011-06-15 EP disclosed
US-20100105653-A1 PYRROLOPYRIMIDINE COMPOUNDS AND THEIR USES NOVARTIS AG 2010-04-29 US disclosed
US-20100105653-A1 PYRROLOPYRIMIDINE COMPOUNDS AND THEIR USES NOVARTIS AG 2010-04-29 US disclosed
US-20100105653-A1 PYRROLOPYRIMIDINE COMPOUNDS AND THEIR USES NOVARTIS AG 2010-04-29 US disclosed
WO-2010020675-A1 PYRROLOPYRIMIDINE COMPOUNDS AS CDK INHIBITORS NOVARTIS AG (CH) 2010-02-25 WO disclosed
WO-2010020675-A1 PYRROLOPYRIMIDINE COMPOUNDS AS CDK INHIBITORS NOVARTIS AG (CH) 2010-02-25 WO disclosed
CN-1980923-A Polycyclic pyridines as potassium ion channel modulators ICAGEN INC (US) 2007-06-13 CN disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (7 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20260146042-A1 PYRROLOPYRIMIDINE COMPOUNDS AND THEIR USES CDK9, CDK6, CDK7 MAPT 3344/4885NR1H2 4468/4885ALDH1A1 3935/4885
US-11261182-B2 Crystal of pyrido[3,4-d]pyrimidine derivative or solvate thereof CDK6, CDK4, CDKL4 MAPT 2457/4885NR1H2 3474/4885ALDH1A1 2897/4885
US-20110152244-A1 PYRROLOPYRIMIDINE COMPOUNDS AND THEIR USES CDK6, CDK8, CDK7 MAPT 2945/4885NR1H2 4214/4885ALDH1A1 3688/4885
US-20230062022-A1 HETEROCYCLIC COMPOUNDS AS KINASE INHIBITORS CDK4, CDK6, CDK8 MAPT 3156/4885NR1H2 4055/4885ALDH1A1 2992/4885
US-20240043428-A1 PYRROLOPYRIMIDINE COMPOUNDS AND THEIR USES CDK6, CDK8, CDK7 MAPT 2945/4885NR1H2 4214/4885ALDH1A1 3688/4885
US-20220296595-A1 CDK INHIBITORS CDKL1, CDK9, CDK6 MAPT 2167/4885NR1H2 2826/4885ALDH1A1 2806/4885
US-20100105653-A1 PYRROLOPYRIMIDINE COMPOUNDS AND THEIR USES CDK6, CDK8, CDK7 MAPT 2945/4885NR1H2 4214/4885ALDH1A1 3688/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.