SCHEMBL2558952

SCHEMBL2558952

COc1cccc(-c2csc(NC(=O)C3CCNCC3)n2)c1

nearest known ligand 0.88

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.88
RAB9A P51151 2/20 0.88
ALDH1A1 P00352 3/20 0.69
HPGD P15428 1/20 0.69
HTT P42858 1/20 0.69
SMN1; SMN2 Q16637 1/20 0.69
HSD17B10 Q99714 1/20 0.69
MEN1 O00255 4/20 0.65
KMT2A Q03164 4/20 0.65
CSNK2A1 P68400 1/20 0.56
ATP4A P20648 2/20 0.55
ATP4B P51164 2/20 0.55
GSK3A P49840 1/20 0.55
GSK3B P49841 1/20 0.55
CDC25A P30304 1/20 0.55
CDC25B P30305 1/20 0.55
CDC25C P30307 1/20 0.55
DUSP3 P51452 1/20 0.55
MAPT P10636 3/20 0.54
THRB P10828 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2560153 0.90 RAB9A (0.70) NPC1RAB9AALDH1A1HPGDHTT
SCHEMBL2559385 0.89 RAB9A (0.69) NPC1RAB9AALDH1A1HPGDHTT
SCHEMBL2553329 0.88 RAB9A (0.67) NPC1RAB9AALDH1A1HPGDHTT
SCHEMBL2562338 0.85 RAB9A (0.63) NPC1RAB9AALDH1A1HPGDHTT
SCHEMBL2558080 0.84 MEN1 (0.68) NPC1RAB9AALDH1A1HPGDHSD17B10
SCHEMBL2557289 0.84 RAB9A (0.61) NPC1RAB9AALDH1A1SMN1; SMN2HSD17B10
SCHEMBL2557829 0.84 RAB9A (0.61) NPC1RAB9AALDH1A1SMN1; SMN2HSD17B10
SCHEMBL2559105 0.84 RAB9A (0.61) NPC1RAB9AALDH1A1HPGDSMN1; SMN2
SCHEMBL2558907 0.84 ABL1 (0.65) NPC1RAB9AALDH1A1SMN1; SMN2MEN1
SCHEMBL2559658 0.83 RAB9A (0.61) NPC1RAB9AALDH1A1HPGDHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011130515-A1 ARYLTHIAZOLYL PIPERIDINES AND RELATED COMPOUNDS AS MODULATORS OF SURVIVAL MOTOR NEURON (SMN) PROTEIN PRODUCTION THE UNITED STATES OF AMERICA, AS REPRESENTED BY THE SECRETARY, DEPARTMENT OF HEALTH AND HUMAN SERVICES (US) 2011-10-20 WO claimed