SCHEMBL2559541

SCHEMBL2559541

CCc1nn(-c2ccc([N+](=O)[O-])cc2)c(C)c1OC(=O)OC

nearest known ligand 0.53

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.53
KDM4E B2RXH2 1/20 0.53
MAPT P10636 9/20 0.47
HTT P42858 2/20 0.47
L3MBTL1 Q9Y468 1/20 0.47
LMNA P02545 4/20 0.45
POLB P06746 2/20 0.44
TDP1 Q9NUW8 1/20 0.44
KMT2A Q03164 1/20 0.44
SLC5A1 P13866 1/20 0.41
SLC5A2 P31639 1/20 0.41
SMN1; SMN2 Q16637 2/20 0.40
RXFP1 Q9HBX9 1/20 0.40
GAA P10253 1/20 0.40
MAPK1 P28482 1/20 0.40
CA9 Q16790 1/20 0.40
PDE4B Q07343 1/20 0.40
PDE4D Q08499 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2561700 0.81 CACNA2D1 (0.44) ALDH1A1KDM4EMAPTPOLBTDP1
SCHEMBL12264807 0.81 MAPT (0.52) ALDH1A1KDM4EMAPTHTTL3MBTL1
SCHEMBL16500135 0.80 ALDH1A1 (0.51) ALDH1A1KDM4EMAPTLMNATDP1
SCHEMBL14482219 0.77 TDP1 (0.54) ALDH1A1KDM4EMAPTHTTL3MBTL1
SCHEMBL16500300 0.69 PDE4B (0.38) ALDH1A1KDM4EMAPTHTTL3MBTL1
SCHEMBL14079407 0.69 NPC1 (0.52) ALDH1A1KDM4EMAPTHTTL3MBTL1
SCHEMBL11041232 0.68 KMT2A (0.49) ALDH1A1KDM4EMAPTHTTL3MBTL1
SCHEMBL2559798 0.68 SLC34A1 (0.49) ALDH1A1KDM4EHTTLMNA
SCHEMBL16692998 0.68 MAPT (0.61) ALDH1A1KDM4EMAPTHTTL3MBTL1
SCHEMBL20037027 0.67 ALDH1A1 (0.75) ALDH1A1KDM4EMAPTHTTL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2552895-B1 PYRAZOLE SYNTHESIS BY COUPLING OF CARBOXYLIC ACID DERIVATIVES AND ENAMINES Westfälische Wilhelms Universität Münster (DE) 2015-02-25 EP disclosed
EP-2552895-A1 PYRAZOLE SYNTHESIS BY COUPLING OF CARBOXYLIC ACID DERIVATIVES AND ENAMINES Westfälische Wilhelms-Universität Münster (DE) 2013-02-06 EP disclosed
WO-2011120861-A1 PYRAZOLE SYNTHESIS BY COUPLING OF CARBOXYLIC ACID DERIVATIVES AND ENAMINES WESTFÄLISHE WILHELMS-UNIVERSITÄT MÜNSTER (DE) 2011-10-06 WO disclosed