SCHEMBL2559968

SCHEMBL2559968

FC(F)(F)Oc1cccc(C2=CCC(Cl)(c3ccc4c(c3)CNCc3nncn3-4)CC2)c1

nearest known ligand 0.37

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
HSD11B1 P28845 1/20 0.37
SCN9A Q15858 1/20 0.31
CYP11B2 P19099 2/20 0.30
CYP11B1 P15538 1/20 0.30
TACR1 P25103 1/20 0.30
BACE1 P56817 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL2558784 0.99 HSD11B1 (0.37) HSD11B1SCN9ACYP11B2
SCHEMBL2563159 0.87 OPRK1 (0.37) CYP11B2CYP11B1
Hydrochloric Acid SCHEMBL2559362 0.86 OPRK1 (0.37) CYP11B2
SCHEMBL2561891 0.84 HSD11B1 (0.36) HSD11B1
Hydrochloric Acid SCHEMBL2558245 0.83 CYP11B2 (0.32) CYP11B2
SCHEMBL2573984 0.81 HSD11B1 (0.35) HSD11B1
Hydrochloric Acid SCHEMBL2545069 0.80 HSD11B1 (0.34) HSD11B1TACR1
SCHEMBL2556274 0.79 CYP11B2 (0.32) CYP11B2CYP11B1
SCHEMBL2559625 0.79 CYP11B2 (0.32) CYP11B2CYP11B1
Hydrochloric Acid SCHEMBL2561790 0.79 CYP11B2 (0.32) CYP11B2CYP11B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2558467-A1 ARYL - /HETEROARYL - CYCLOHEXENYL - TETRAAZABENZO [E]AZULENES AS VASOPRESSIN ANTAGONISTS F. Hoffmann-La Roche AG (CH) 2013-02-20 EP claimed
WO-2011128265-A1 ARYL - /HETEROARYL - CYCLOHEXENYL - TETRAAZABENZO [E] AZULENES AS VASOPRESSIN ANTAGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2011-10-20 WO claimed
EP-2558467-A1 ARYL - /HETEROARYL - CYCLOHEXENYL - TETRAAZABENZO [E]AZULENES AS VASOPRESSIN ANTAGONISTS F. Hoffmann-La Roche AG (CH) 2013-02-20 EP disclosed
WO-2011128265-A1 ARYL - /HETEROARYL - CYCLOHEXENYL - TETRAAZABENZO [E] AZULENES AS VASOPRESSIN ANTAGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2011-10-20 WO disclosed