SCHEMBL2556274

SCHEMBL2556274

Fc1cccnc1C1=CCC(Cl)(c2ccc3c(c2)CNCc2nncn2-3)CC1

nearest known ligand 0.33

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
CYP11B2 P19099 2/20 0.32
CYP11B1 P15538 1/20 0.32
TRPV1 Q8NER1 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL2561790 0.85 CYP11B2 (0.32) CYP11B2CYP11B1
SCHEMBL2563159 0.84 OPRK1 (0.37) CYP11B2CYP11B1
SCHEMBL2560463 0.84
Hydrochloric Acid SCHEMBL2558245 0.84 CYP11B2 (0.32) CYP11B2
Hydrochloric Acid SCHEMBL2559362 0.83 OPRK1 (0.37) CYP11B2
SCHEMBL2563129 0.83 TRPV1 (0.34) CYP11B2CYP11B1TRPV1
Hydrochloric Acid SCHEMBL2551927 0.80 OPRK1 (0.31)
SCHEMBL2564607 0.79 AVPR1A (0.35) CYP11B2CYP11B1
SCHEMBL2574177 0.79 GRM5 (0.38) TRPV1
SCHEMBL2559968 0.79 HSD11B1 (0.37) CYP11B2CYP11B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2558467-A1 ARYL - /HETEROARYL - CYCLOHEXENYL - TETRAAZABENZO [E]AZULENES AS VASOPRESSIN ANTAGONISTS F. Hoffmann-La Roche AG (CH) 2013-02-20 EP disclosed
WO-2011128265-A1 ARYL - /HETEROARYL - CYCLOHEXENYL - TETRAAZABENZO [E] AZULENES AS VASOPRESSIN ANTAGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2011-10-20 WO disclosed