SCHEMBL2559970

SCHEMBL2559970

COc1ccc(C=O)c2c1oc1cnccc12

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 2/20 0.39
TDO2 P48775 2/20 0.39
ERN1 O75460 3/20 0.36
CYP17A1 P05093 1/20 0.36
CYP19A1 P11511 1/20 0.36
CYP11B1 P15538 1/20 0.36
CYP11B2 P19099 1/20 0.36
CYP1A1 P04798 3/20 0.36
CYP1B1 Q16678 3/20 0.36
PDE4A P27815 2/20 0.36
PDE4B Q07343 2/20 0.36
PDE4C Q08493 2/20 0.36
PDE4D Q08499 2/20 0.36
CHUK O15111 1/20 0.36
PRKD3 O94806 1/20 0.36
PRKCG P05129 1/20 0.36
PRKCB P05771 1/20 0.36
PRKCA P17252 1/20 0.36
CSNK2A2 P19784 1/20 0.36
PRKCH P24723 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2556718 0.90 CYP17A1 (0.39) ERN1CYP17A1CYP19A1CYP11B1CYP11B2
SCHEMBL2556489 0.86 CYP19A1 (0.40) CYP19A1CYP11B1CYP11B2ALDH1A1MAPT
SCHEMBL2556065 0.84 PDE4B (0.43) IDO1TDO2CYP17A1CYP19A1CYP11B1
SCHEMBL2562773 0.83 HPGD (0.41) IDO1TDO2CYP1A1CYP1B1PDE4A
SCHEMBL2560821 0.83 HPGD (0.41) IDO1TDO2CYP1A1CYP1B1PDE4A
SCHEMBL1647979 0.81 MAOA (0.52) CYP17A1CYP19A1CYP11B1CYP11B2PDE4B
SCHEMBL2560102 0.80 ERN1 (0.43) IDO1TDO2ERN1CYP17A1CYP19A1
SCHEMBL2556731 0.79 CCNC (0.42) CYP1A1CYP1B1CYP1A2MAPTLMNA
SCHEMBL13233338 0.76 PDE4A (0.36) PDE4APDE4BPDE4CPDE4D
SCHEMBL3724543 0.75 MAOA (0.57) CYP17A1CYP19A1CYP11B1CYP11B2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011132051-A2 TRICYCLE COMPOUNDS AS PHOSPHODIESTERASE-10 INHIBITORS GLENMARK PHARMACEUTICALS S.A. (CH) 2011-10-27 WO disclosed