Ethaverine

Ethaverine

SCHEMBL25606

CCOc1ccc(Cc2nccc3cc(OCC)c(OCC)cc23)cc1OCC

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE3A Q14432 10/20 1.00
SMN1; SMN2 Q16637 5/20 1.00
CYP3A4 P08684 4/20 1.00
MAPK1 P28482 4/20 1.00
LMNA P02545 3/20 1.00
CYP1A2 P05177 2/20 1.00
CYP2C9 P11712 2/20 1.00
TSHR P16473 2/20 1.00
PDE4A P27815 2/20 1.00
KCNH2 Q12809 2/20 1.00
TDP1 Q9NUW8 2/20 1.00
MEN1 O00255 1/20 1.00
ADRA2A P08913 1/20 1.00
ADORA3 P0DMS8 1/20 1.00
CHRM1 P11229 1/20 1.00
DRD1 P21728 1/20 1.00
TBXA2R P21731 1/20 1.00
ADRA1A P35348 1/20 1.00
DRD3 P35462 1/20 1.00
KMT2A Q03164 1/20 1.00

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Ethaverine SCHEMBL29355739 1.00 PDE3A (1.00) PDE3ASMN1; SMN2CYP3A4MAPK1LMNA
Ethaverine SCHEMBL29500886 1.00 PDE3A (1.00) PDE3ASMN1; SMN2CYP3A4MAPK1LMNA
Ethaverine SCHEMBL29624566 0.99 SMN1; SMN2 (1.00) PDE3ASMN1; SMN2CYP3A4MAPK1LMNA
Ethaverine SCHEMBL9614397 0.99 SMN1; SMN2 (1.00) PDE3ASMN1; SMN2CYP3A4MAPK1LMNA
Ethaverine SCHEMBL16180359 0.99 SMN1; SMN2 (1.00) PDE3ASMN1; SMN2CYP3A4MAPK1LMNA
Ethaverine SCHEMBL317507 0.99 SMN1; SMN2 (1.00) PDE3ASMN1; SMN2CYP3A4MAPK1LMNA
Ethaverine SCHEMBL30417501 0.99 SMN1; SMN2 (1.00) PDE3ASMN1; SMN2CYP3A4MAPK1LMNA
Ethaverine SCHEMBL17603566 0.99 PDE3A (0.97) PDE3ASMN1; SMN2CYP3A4MAPK1LMNA
SCHEMBL2455134 0.93 PDE3A (0.87) PDE3ASMN1; SMN2CYP3A4MAPK1LMNA
SCHEMBL2460329 0.91 PDE3A (0.83) PDE3ASMN1; SMN2CYP3A4MAPK1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1004 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230233483-A1 COMPOUND AND METHOD FOR THE TREATMENT OF CORONAVIRUSES APTEEUS (FR) 2023-07-27 US claimed
US-20230126310-A1 COMPOSITIONS FOR CORONAVIRUS INFECTION TREATMENT AND/OR PREVENTION FRAUNHOFER GES FORSCHUNG (DE) 2023-04-27 US claimed
EP-4126234-A1 COMPOSITIONS FOR CORONAVIRUS INFECTION TREATMENT AND/OR PREVENTION Fraunhofer-Gesellschaft zur Förderung der angewandten Forschung e.V. (DE) 2023-02-08 EP claimed
WO-2022164850-A1 COMPOUNDS TO PREVENT OR TREAT SARS-CoV-2 VARIANT INFECTION UNIVERSITY OF FLORIDA RESEARCH FOUNDATION, INCORPORATED (US) 2022-08-04 WO claimed
WO-2021198440-A1 COMPOSITIONS FOR CORONAVIRUS INFECTION TREATMENT AND/OR PREVENTION Fraunhofer-Gesellschaft zur Förderung der angewandten Forschung e.V. (DE) 2021-10-07 WO claimed
WO-2021054927-A2 GLUTATHIONE-CHOLESTEROL DERIVATIVES AS BRAIN TARGETING AGENTS SOUTH DAKOTA BOARD OF REGENTS (US) 2021-03-25 WO claimed
EP-3635130-A1 PRECISION MEDICINE FOR TREATING AND PREVENTING SUICIDALITY Indiana University Research and Technology Corporation (US) 2020-04-15 EP claimed
US-20200048305-A1 GLUTATHIONE-CHOLESTEROL DERIVATIVES AS BRAIN TARGETING AGENTS SOUTH DAKOTA BOARD OF REGENTS (US) 2020-02-13 US claimed
WO-2018209341-A1 PRECISION MEDICINE FOR TREATING AND PREVENTING SUICIDALITY INDIANA UNIVERSITY RESEARCH AND TECHNOLOGY CORPORATION (US) 2018-11-15 WO claimed
US-20170269060-A1 Assays and Compounds to Treat Kidney Diseases RUSH UNIVERSITY MEDICAL CENTER (US) 2017-09-21 US claimed
WO-2002039952-A2 SYNERGISTIC ECTA COMPOSITIONS NEWBIOTICS, INC. (US) 2002-05-23 WO claimed
CN-1294519-A Pharmaceutical composition containing a compound having an activity of promoting the absorption of an active ingredient INPHARMA SA (CH) 2001-05-09 CN claimed
EP-1073470-A1 PHARMACEUTICAL COMPOSITIONS CONTAINING COMPOUNDS WITH ACTIVITY FOR THE ENHANCEMENT OF ABSORPTION OF ACTIVE INGREDIENTS INPHARMA S.A. (CH) 2001-02-07 EP claimed
WO-2000048636-A1 PHARMACEUTICAL COMPOSITIONS CONTAINING COMPOUNDS WITH ACTIVITY FOR THE ENHANCEMENT OF ABSORPTION OF ACTIVE INGREDIENTS INPHARMA S.A. (CH) 2000-08-24 WO claimed
US-5491051-A HAVING LIGHT SENSITIVE LAYER, TRANSPARENT MAGNETIC RECORDING LAYER CONTAINING TRANSPARENT BINDER, FERROMAGNETIC PARTICLES, ABRASIVE PARTICLES WITH SPECIFIED PROPERTIES; DURABILITY EASTMAN KODAK COMPANY (US) 1996-02-13 US claimed
US-5256652-A Administering peripheral vasodilator and hydroxy-B-cyclo-dextrin to enhance erection PHARMEDIC CO. (US) 1993-10-26 US claimed
WO-1992003141-A1 TOPICAL COMPOSITIONS AND METHODS FOR TREATMENT OF MALE IMPOTENCE PHARMEDIC CO. (US) 1992-03-05 WO claimed
US-5026544-A Administering papaverine compound with interferon BOARD OF REAGENTS, THE UNIVERSITY OF TEXAS SYSTEM (US) 1991-06-25 US claimed
US-4849412-A PAPAVERINE COMPOUND, NUCLEOSIDE ANALOG BOARD OF REGENTS, THE UNIVERSITY OF TEXAS SYSTEM (US) 1989-07-18 US claimed
WO-1987007508-A1 METHODS AND COMPOSITIONS FOR TREATING VIRAL INFECTIONS BOARD OF REGENTS, THE UNIVERSITY OF TEXAS SYSTEM (US) 1987-12-17 WO claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20200048305-A1 GLUTATHIONE-CHOLESTEROL DERIVATIVES AS BRAIN TARGETING AGENTS GSTK1, GSTO1, GSTM2 PDE3A 1351/4885SMN1; SMN2 4125/4885CYP3A4 2149/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.