SCHEMBL2561201

SCHEMBL2561201

COC(=O)Oc1c(-c2ncccc2C)nn(-c2ccccc2)c1C

nearest known ligand 0.42

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 3/20 0.42
KMT2A Q03164 3/20 0.42
ALDH1A1 P00352 5/20 0.41
TSHR P16473 1/20 0.40
RAB9A P51151 5/20 0.40
MAPT P10636 3/20 0.40
NPSR1 Q6W5P4 1/20 0.40
P2RX7 Q99572 1/20 0.40
NPC1 O15118 4/20 0.40
MAPK1 P28482 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
HPGD P15428 1/20 0.38
PDE4D Q08499 1/20 0.38
HTT P42858 2/20 0.37
LMNA P02545 1/20 0.37
POLB P06746 1/20 0.37
ATM Q13315 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2553897 0.83 MEN1 (0.58) MEN1KMT2AALDH1A1TSHRRAB9A
SCHEMBL14553212 0.81 MEN1 (0.52) MEN1KMT2AALDH1A1TSHRRAB9A
SCHEMBL12264900 0.78 MEN1 (0.66) MEN1KMT2AALDH1A1RAB9AMAPT
SCHEMBL2557760 0.77 MEN1 (0.48) MEN1KMT2AALDH1A1RAB9AMAPT
SCHEMBL2557260 0.77 KDM4E (0.48) MEN1KMT2AALDH1A1TSHRRAB9A
SCHEMBL2557580 0.77 KMT2A (0.48) MEN1KMT2AALDH1A1TSHRRAB9A
SCHEMBL2560863 0.75 ALDH1A1 (0.55) MEN1KMT2AALDH1A1NPSR1SMN1; SMN2
SCHEMBL2576433 0.74 TSHR (0.47) MEN1KMT2AALDH1A1TSHRRAB9A
SCHEMBL16500084 0.73 TSHR (0.43) MEN1KMT2AALDH1A1TSHRRAB9A
SCHEMBL16500135 0.72 ALDH1A1 (0.51) MEN1KMT2AALDH1A1RAB9AMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2552895-B1 PYRAZOLE SYNTHESIS BY COUPLING OF CARBOXYLIC ACID DERIVATIVES AND ENAMINES Westfälische Wilhelms Universität Münster (DE) 2015-02-25 EP disclosed
EP-2552895-A1 PYRAZOLE SYNTHESIS BY COUPLING OF CARBOXYLIC ACID DERIVATIVES AND ENAMINES Westfälische Wilhelms-Universität Münster (DE) 2013-02-06 EP disclosed
WO-2011120861-A1 PYRAZOLE SYNTHESIS BY COUPLING OF CARBOXYLIC ACID DERIVATIVES AND ENAMINES WESTFÄLISHE WILHELMS-UNIVERSITÄT MÜNSTER (DE) 2011-10-06 WO disclosed