SCHEMBL2557760

SCHEMBL2557760

COC(=O)Oc1c(-c2cccc(C)c2)nn(-c2ccccc2)c1C

nearest known ligand 0.48

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 3/20 0.48
KMT2A Q03164 3/20 0.48
MAPT P10636 3/20 0.46
TP53 P04637 2/20 0.46
LMNA P02545 5/20 0.46
ALDH1A1 P00352 8/20 0.46
GRM5 P41594 1/20 0.44
RPA1 P27694 1/20 0.44
NPC1 O15118 1/20 0.43
NFKB1 P19838 1/20 0.43
RAB9A P51151 1/20 0.43
NFKB2 Q00653 1/20 0.43
RELA Q04206 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
KCNJ6 P48051 1/20 0.42
KCNJ5 P48544 1/20 0.42
KCNJ3 P48549 1/20 0.42
KDM4E B2RXH2 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2553897 0.90 MEN1 (0.58) MEN1KMT2AMAPTLMNAALDH1A1
SCHEMBL2560863 0.82 ALDH1A1 (0.55) MEN1KMT2AALDH1A1GRM5SMN1; SMN2
SCHEMBL2557580 0.81 KMT2A (0.48) MEN1KMT2AMAPTTP53LMNA
SCHEMBL12264907 0.81 MEN1 (0.62) MEN1KMT2AMAPTTP53LMNA
SCHEMBL16500135 0.79 ALDH1A1 (0.51) MEN1KMT2AMAPTLMNAALDH1A1
SCHEMBL2554340 0.78 KMT2A (0.56) MEN1KMT2AMAPTTP53ALDH1A1
SCHEMBL14482936 0.78 MEN1 (0.79) MEN1KMT2AMAPTTP53LMNA
SCHEMBL2561201 0.77 MEN1 (0.42) MEN1KMT2AMAPTLMNAALDH1A1
SCHEMBL2557260 0.77 KDM4E (0.48) MEN1KMT2AMAPTLMNAALDH1A1
SCHEMBL16500067 0.75 TP53 (0.48) MEN1KMT2AMAPTTP53LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2552895-B1 PYRAZOLE SYNTHESIS BY COUPLING OF CARBOXYLIC ACID DERIVATIVES AND ENAMINES Westfälische Wilhelms Universität Münster (DE) 2015-02-25 EP disclosed
EP-2552895-A1 PYRAZOLE SYNTHESIS BY COUPLING OF CARBOXYLIC ACID DERIVATIVES AND ENAMINES Westfälische Wilhelms-Universität Münster (DE) 2013-02-06 EP disclosed
WO-2011120861-A1 PYRAZOLE SYNTHESIS BY COUPLING OF CARBOXYLIC ACID DERIVATIVES AND ENAMINES WESTFÄLISHE WILHELMS-UNIVERSITÄT MÜNSTER (DE) 2011-10-06 WO disclosed