SCHEMBL2562269

SCHEMBL2562269

Cc1cc(-c2nc3ccccc3c(=O)n2-c2ccc(N3CCOCC3)cc2)cc(C)c1OCCO

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
JUN P05412 1/20 0.51
NFKB1 P19838 1/20 0.51
NFKB2 Q00653 1/20 0.51
RELA Q04206 1/20 0.51
AHR P35869 1/20 0.48
MAPT P10636 5/20 0.48
KCNH2 Q12809 2/20 0.48
HRH3 Q9Y5N1 2/20 0.48
ALDH1A1 P00352 9/20 0.48
RAB9A P51151 2/20 0.48
KDM4E B2RXH2 2/20 0.48
NPC1 O15118 1/20 0.48
HCRTR1 O43613 1/20 0.48
LMNA P02545 1/20 0.48
GAA P10253 1/20 0.48
TDO2 P48775 1/20 0.46
IDO2 Q6ZQW0 1/20 0.46
SYK P43405 1/20 0.45
ADRA1A P35348 1/20 0.45
NPSR1 Q6W5P4 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2561941 0.85 ALDH1A1 (0.51) MAPTKCNH2HRH3ALDH1A1RAB9A
SCHEMBL2566454 0.85 ALDH1A1 (0.51) MAPTKCNH2HRH3ALDH1A1RAB9A
SCHEMBL2565658 0.85 SMN1; SMN2 (0.52) JUNNFKB1NFKB2RELAMAPT
SCHEMBL2562815 0.85 ALDH1A1 (0.51) MAPTKCNH2HRH3ALDH1A1RAB9A
SCHEMBL2564148 0.85 ALDH1A1 (0.51) MAPTKCNH2HRH3ALDH1A1RAB9A
SCHEMBL15512657 0.85 MAPK1 (0.57) MAPTKCNH2HRH3ALDH1A1RAB9A
SCHEMBL2562510 0.84 ALDH1A1 (0.49) MAPTKCNH2HRH3ALDH1A1RAB9A
SCHEMBL2565762 0.84 ALDH1A1 (0.49) MAPTKCNH2HRH3ALDH1A1RAB9A
SCHEMBL2562976 0.84 ALDH1A1 (0.49) MAPTKCNH2HRH3ALDH1A1RAB9A
SCHEMBL2567691 0.84 ALDH1A1 (0.49) MAPTKCNH2HRH3ALDH1A1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 28 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8952021-B2 Compounds for the prevention and treatment of cardiovascular disease RESVERLOGIX CORP. (CA) 2015-02-10 US claimed
EP-2382194-B1 COMPOUNDS FOR THE PREVENTION AND TREATMENT OF CARDIOVASCULAR DISEASE RESVERLOGIX CORP (CA) 2014-03-12 EP claimed
US-20110294807-A1 COMPOUNDS FOR THE PREVENTION AND TREATMENT OF CARDIOVASCULAR DISEASE RESVERLOGIX CORP. (CA) 2011-12-01 US claimed
EP-2382194-A2 COMPOUNDS FOR THE PREVENTION AND TREATMENT OF CARDIOVASCULAR DISEASE RESVERLOGIX CORP. (CA) 2011-11-02 EP claimed
WO-2010079431-A2 COMPOUNDS FOR THE PREVENTION AND TREATMENT OF CARDIOVASCULAR DISEASE RESVERLOGIX CORP. (CA) 2010-07-15 WO claimed
WO-2015081284-A1 BIVALENT BROMODOMAIN LIGANDS, AND METHODS OF USING SAME COFERON, INC. (US) 2015-06-04 WO disclosed
WO-2015081280-A1 BROMODOMAIN LIGANDS CAPABLE OF DIMERIZING IN AN AQUEOUS SOLUTION COFERON, INC. (US) 2015-06-04 WO disclosed
EP-2660238-B1 Compounds for the prevention and treatment of cardiovascular disease RESVERLOGIX CORP (CA) 2015-05-06 EP disclosed
EP-2660238-B1 Compounds for the prevention and treatment of cardiovascular disease RESVERLOGIX CORP (CA) 2015-05-06 EP disclosed
US-8952021-B2 Compounds for the prevention and treatment of cardiovascular disease RESVERLOGIX CORP. (CA) 2015-02-10 US disclosed
US-8952021-B2 Compounds for the prevention and treatment of cardiovascular disease RESVERLOGIX CORP. (CA) 2015-02-10 US disclosed
US-8952021-B2 Compounds for the prevention and treatment of cardiovascular disease RESVERLOGIX CORP. (CA) 2015-02-10 US disclosed
WO-2013033268-A2 BIVALENT BROMODOMAIN LIGANDS, AND METHODS OF USING SAME COFERON, INC. (US) 2013-03-07 WO disclosed
WO-2013033269-A1 BIOORTHOGONAL MONOMERS CAPABLE OF DIMERIZING AND TARGETING BROMODOMAINS AND METHODS OF USING SAME COFERON, INC. (US) 2013-03-07 WO disclosed
US-20110294807-A1 COMPOUNDS FOR THE PREVENTION AND TREATMENT OF CARDIOVASCULAR DISEASE RESVERLOGIX CORP. (CA) 2011-12-01 US disclosed
US-20110294807-A1 COMPOUNDS FOR THE PREVENTION AND TREATMENT OF CARDIOVASCULAR DISEASE RESVERLOGIX CORP. (CA) 2011-12-01 US disclosed
US-20110294807-A1 COMPOUNDS FOR THE PREVENTION AND TREATMENT OF CARDIOVASCULAR DISEASE RESVERLOGIX CORP. (CA) 2011-12-01 US disclosed
EP-2382194-A2 COMPOUNDS FOR THE PREVENTION AND TREATMENT OF CARDIOVASCULAR DISEASE RESVERLOGIX CORP. (CA) 2011-11-02 EP disclosed
WO-2010079431-A2 COMPOUNDS FOR THE PREVENTION AND TREATMENT OF CARDIOVASCULAR DISEASE RESVERLOGIX CORP. (CA) 2010-07-15 WO disclosed
WO-2010079431-A2 COMPOUNDS FOR THE PREVENTION AND TREATMENT OF CARDIOVASCULAR DISEASE RESVERLOGIX CORP. (CA) 2010-07-15 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110294807-A1 COMPOUNDS FOR THE PREVENTION AND TREATMENT OF CARDIOVASCULAR DISEASE APOB, APOL1, LDLR JUN 768/4885NFKB1 505/4885NFKB2 650/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.