SCHEMBL25650490

SCHEMBL25650490

O=C(O)c1nnc(-n2ccnc2)s1

nearest known ligand 0.43

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ADH5 P11766 8/20 0.43
ENPP2 Q13822 1/20 0.40
MKNK1 Q9BUB5 1/20 0.40
MKNK2 Q9HBH9 1/20 0.40
TBXAS1 P24557 3/20 0.39
CYP3A4 P08684 2/20 0.38
BAZ2B Q9UIF8 1/20 0.38
IDO1 P14902 2/20 0.38
STING1 Q86WV6 1/20 0.36
HTT P42858 1/20 0.36
HTR2A P28223 1/20 0.35
HTR2C P28335 1/20 0.35
HTR2B P41595 1/20 0.35
MEN1 O00255 1/20 0.34
ALOX15 P16050 1/20 0.34
TSHR P16473 1/20 0.34
KMT2A Q03164 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25650489 0.79 OGA (0.44) TBXAS1CYP3A4BAZ2BHTTMEN1
SCHEMBL25650245 0.75 STING1 (0.64) CYP3A4STING1
SCHEMBL25650246 0.72 STING1 (0.57) STING1
SCHEMBL8150666 0.72 LMNA (0.44) ENPP2MKNK1MKNK2CYP3A4IDO1
SCHEMBL18114204 0.70 PIK3CD (0.48) ADH5TBXAS1CYP3A4BAZ2BHTT
SCHEMBL31216537 0.69 CHEK1 (0.48) ADH5
SCHEMBL31216541 0.69 ADH5 (0.42) ADH5ENPP2MKNK1MKNK2TBXAS1
SCHEMBL7020662 0.66 DAO (0.35) TSHR
SCHEMBL28766887 0.65 ADH5 (0.47) ADH5ENPP2MKNK1MKNK2CYP3A4
SCHEMBL2628931 0.65 CYP3A4 (0.39) ENPP2MKNK1MKNK2CYP3A4IDO1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023103850-A1 SMALL MOLECULE STING AGONIST, PREPARATION METHOD THEREFOR, AND APPLICATION 中国科学院上海药物研究所 2023-06-15 WO disclosed