SCHEMBL2568952

SCHEMBL2568952

COC(=O)c1ccc2c(c1)CC(C)(C)C(c1ccc(NCC(C)C)cc1)N2

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CRBN Q96SW2 1/20 0.39
SMN1; SMN2 Q16637 3/20 0.38
ALDH1A1 P00352 3/20 0.38
MEN1 O00255 2/20 0.38
KMT2A Q03164 2/20 0.38
RAB9A P51151 3/20 0.38
NPC1 O15118 2/20 0.38
MAPT P10636 4/20 0.37
AR P10275 1/20 0.36
POLB P06746 2/20 0.36
HSD17B10 Q99714 1/20 0.36
NAMPT P43490 1/20 0.36
CA1 P00915 2/20 0.35
CA2 P00918 2/20 0.35
KDM4E B2RXH2 3/20 0.35
TP53 P04637 1/20 0.35
MDM2 Q00987 1/20 0.35
MAPK1 P28482 2/20 0.35
FNTA P49354 1/20 0.35
FNTB P49356 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2574265 0.90 HCAR3 (0.38) ALDH1A1MEN1KMT2AMAPTPOLB
SCHEMBL2589366 0.86 SMN1; SMN2 (0.38) CRBNSMN1; SMN2ALDH1A1MEN1KMT2A
SCHEMBL2576665 0.86 ALDH1A1 (0.39) SMN1; SMN2ALDH1A1MEN1KMT2ARAB9A
SCHEMBL2529286 0.85 ALDH1A1 (0.41) CRBNSMN1; SMN2ALDH1A1MEN1KMT2A
SCHEMBL2575481 0.83 CRBN (0.45) CRBNSMN1; SMN2ALDH1A1MEN1KMT2A
SCHEMBL2531931 0.82 ALDH1A1 (0.42) CRBNSMN1; SMN2ALDH1A1MEN1KMT2A
SCHEMBL2572744 0.81 ITGB3 (0.40) SMN1; SMN2ALDH1A1MEN1KMT2ARAB9A
SCHEMBL2535710 0.80 PTPN1 (0.49) SMN1; SMN2ALDH1A1MEN1KMT2ARAB9A
SCHEMBL2531914 0.80 POLB (0.44) SMN1; SMN2ALDH1A1MEN1KMT2ARAB9A
SCHEMBL2527699 0.80 MAPT (0.42) SMN1; SMN2ALDH1A1MEN1KMT2ARAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2558449-A1 NOVEL 3,3-DIMETHYL TETRAHYDROQUINOLINE DERIVATIVES F. Hoffmann-La Roche AG (CH) 2013-02-20 EP disclosed
WO-2011128251-A1 NOVEL 3,3-DIMETHYL TETRAHYDROQUINOLINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2011-10-20 WO disclosed