SCHEMBL2569708

SCHEMBL2569708

CN1CCc2ccc(NC(=O)[C@@H](CNC(=O)c3ccccc3)NC(=O)Oc3ccc(Cl)s3)cc2CC1

nearest known ligand 0.39

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 16/20 0.39
CYP3A4 P08684 1/20 0.39
NPC1 O15118 1/20 0.39
TP53 P04637 1/20 0.39
GAA P10253 1/20 0.39
NFKB1 P19838 1/20 0.39
HTT P42858 1/20 0.39
RAB9A P51151 1/20 0.39
NFKB2 Q00653 1/20 0.39
RELA Q04206 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
ROCK1 Q13464 2/20 0.38
TMPRSS2 O15393 1/20 0.37
PRMT5 O14744 1/20 0.37
WDR77 Q9BQA1 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2571141 0.92 CCKBR (0.38) ROCK2CYP3A4NPC1TP53GAA
SCHEMBL2563392 0.90 ROCK2 (0.39) ROCK2CYP3A4NPC1TP53GAA
SCHEMBL2572758 0.89 F10 (0.35) ROCK2CYP3A4
SCHEMBL3380237 0.89 CCKBR (0.35) ROCK2
SCHEMBL2569493 0.88 PSEN1 (0.41)
SCHEMBL3036150 0.88 F10 (0.46) ROCK2TMPRSS2
SCHEMBL2565436 0.87 CCKBR (0.38) ROCK2HTT
SCHEMBL3378613 0.87 DRD2 (0.35) ROCK2NPC1RAB9A
SCHEMBL2566646 0.87 MAPT (0.42)
SCHEMBL2580055 0.86 CA1 (0.40) ROCK2NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1899330-B9 SUBSTITUTED GLYCINAMIDES HAVING AN ANTITHROMBOTIC AND FACTOR XA-INHIBITING EFFECT BOEHRINGER INGELHEIM INT (DE) 2011-11-09 EP disclosed
EP-1899330-B1 SUBSTITUTED GLYCINAMIDES HAVING AN ANTITHROMBOTIC AND FACTOR XA-INHIBITING EFFECT BOEHRINGER INGELHEIM INT (DE) 2010-11-24 EP disclosed