SCHEMBL25700511

SCHEMBL25700511

Fc1ccc(-c2nc3cnc4[nH]ccc4c3[nH]2)cc1F

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2C8 P10632 1/20 0.41
TGFBR1 P36897 1/20 0.41
RPS6KA3 P51812 4/20 0.40
DYRK1A Q13627 2/20 0.40
FLT3 P36888 2/20 0.40
AURKA O14965 1/20 0.40
DAPK3 O43293 1/20 0.40
JAK2 O60674 1/20 0.40
PRKD3 O94806 1/20 0.40
MAP4K4 O95819 1/20 0.40
PAK4 O96013 1/20 0.40
NTRK1 P04629 1/20 0.40
CSF1R P07333 1/20 0.40
RET P07949 1/20 0.40
IGF1R P08069 1/20 0.40
MET P08581 1/20 0.40
PIM1 P11309 1/20 0.40
FGFR1 P11362 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25697123 0.85 MAPK1 (0.50) RPS6KA3METKDRTRPA1MAPK1
SCHEMBL25696459 0.80 MAPK1 (0.48) RPS6KA3DYRK1ADAPK3JAK2PRKD3
SCHEMBL25696601 0.80 TNKS (0.46) AURKAJAK2KDRKCNH2
SCHEMBL20290060 0.80 JAK1 (0.44) RPS6KA3AURKAJAK2KDRJAK3
SCHEMBL25696739 0.79 NPC1 (0.49) CYP1A2CYP3A4TGFBR1RPS6KA3DYRK1A
SCHEMBL27432231 0.79 HSD17B1 (0.44) JAK2MAPK1
SCHEMBL20289959 0.77 JAK1 (0.41) CYP3A4DYRK1AAURKAJAK2KDR
SCHEMBL25697037 0.77 CCNT1 (0.38) AURKAJAK2PRKD3MAP4K4RET
SCHEMBL25696885 0.77 MAPK1 (0.53) AURKAJAK2JAK3TBK1MAPK1
SCHEMBL27432272 0.77 AMY1A (0.39) RPS6KA3DYRK1AFLT3FGFR1DYRK1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4393923-A1 PYRIDO RING COMPOUND, PREPARATION METHOD THEREFOR, INTERMEDIATE, COMPOSITION, AND APPLICATION Yiyou Biotech (Shanghai) Co., Ltd. (CN) 2024-07-03 EP disclosed
WO-2023115327-A1 PYRIDO RING COMPOUND, PREPARATION METHOD THEREFOR, INTERMEDIATE, COMPOSITION, AND APPLICATION 中国药科大学 2023-06-29 WO disclosed