SCHEMBL257153

SCHEMBL257153

CCS(=O)(=O)c1ccc(CC(=O)OC)cc1

nearest known ligand 0.58

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
MMP9 P14780 1/20 0.57
CYP4F2 P78329 1/20 0.56
CYP4A11 Q02928 1/20 0.56
RORC P51449 11/20 0.53
PSIP1 O75475 1/20 0.52
ALDH1A1 P00352 3/20 0.49
GAA P10253 2/20 0.49
KDM4E B2RXH2 1/20 0.49
NPC1 O15118 1/20 0.49
HPGD P15428 1/20 0.49
RAB9A P51151 1/20 0.49
SMN1; SMN2 Q16637 1/20 0.49
CTSG P08311 1/20 0.47
CMA1 P23946 1/20 0.47
GFER P55789 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL175501 0.85 CYP4F2 (0.60) MMP9CYP4F2CYP4A11ALDH1A1GAA
SCHEMBL2665972 0.84 KMT2A (0.57) RORCPSIP1ALDH1A1GAAKDM4E
SCHEMBL1096091 0.84 CYP4F2 (0.58) MMP9CYP4F2CYP4A11ALDH1A1GAA
SCHEMBL30898772 0.83 IDO1 (0.56) CYP4F2CYP4A11RORCPSIP1ALDH1A1
SCHEMBL4113212 0.82 CYP4F2 (0.76) CYP4F2CYP4A11ALDH1A1GAAKDM4E
SCHEMBL23174344 0.82 MMP9 (0.64) MMP9CYP4F2CYP4A11RORCALDH1A1
SCHEMBL167112 0.82 MMP9 (0.51) MMP9CYP4F2CYP4A11RORCALDH1A1
SCHEMBL10141348 0.82 CYP4F2 (0.56) MMP9CYP4F2CYP4A11ALDH1A1GAA
SCHEMBL22664337 0.82 CA2 (0.58) CYP4F2CYP4A11ALDH1A1GAAKDM4E
SCHEMBL184666 0.82 CYP4F2 (0.56) MMP9CYP4F2CYP4A11ALDH1A1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021228215-A1 BIARYL COMPOUND CAPABLE OF SERVING AS RORγ REGULATOR 上海辉启生物医药科技有限公司 2021-11-18 WO disclosed
WO-2012028100-A1 NOVEL COMPOUNDS GLAXO GROUP LIMITED (GB) 2012-03-08 WO disclosed