SCHEMBL184666

SCHEMBL184666

COC(=O)Cc1ccc(S(=O)(=O)Cl)cc1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP4F2 P78329 1/20 0.56
CYP4A11 Q02928 1/20 0.56
MMP9 P14780 1/20 0.50
ALDH1A1 P00352 4/20 0.49
NPC1 O15118 3/20 0.49
RAB9A P51151 3/20 0.49
SMN1; SMN2 Q16637 5/20 0.49
GAA P10253 2/20 0.49
KDM4E B2RXH2 1/20 0.49
HPGD P15428 1/20 0.49
CTSG P08311 1/20 0.47
CMA1 P23946 1/20 0.47
GFER P55789 1/20 0.46
HSP90AB1 P08238 1/20 0.46
HTT P42858 1/20 0.45
EGFR P00533 1/20 0.44
ERBB2 P04626 1/20 0.44
CA12 O43570 1/20 0.44
CA1 P00915 1/20 0.44
CA2 P00918 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1096091 0.84 CYP4F2 (0.58) CYP4F2CYP4A11MMP9ALDH1A1NPC1
SCHEMBL119585 0.83 LMNA (0.54) CYP4F2CYP4A11ALDH1A1SMN1; SMN2GAA
SCHEMBL343527 0.83 IDO1 (0.56) CYP4F2CYP4A11ALDH1A1NPC1RAB9A
SCHEMBL4113212 0.82 CYP4F2 (0.76) CYP4F2CYP4A11ALDH1A1NPC1RAB9A
SCHEMBL257153 0.82 MMP9 (0.57) CYP4F2CYP4A11MMP9ALDH1A1NPC1
SCHEMBL10141348 0.82 CYP4F2 (0.56) CYP4F2CYP4A11MMP9ALDH1A1NPC1
SCHEMBL22664337 0.82 CA2 (0.58) CYP4F2CYP4A11ALDH1A1SMN1; SMN2GAA
SCHEMBL16092814 0.82 CYP4F2 (0.56) CYP4F2CYP4A11MMP9ALDH1A1NPC1
SCHEMBL8934772 0.81 MTNR1A (0.42) CYP4F2CYP4A11MMP9ALDH1A1KDM4E
SCHEMBL12440455 0.81 ALDH1A1 (0.60) CYP4F2CYP4A11ALDH1A1NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 90 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230357214-A1 NOVEL LXR MODULATORS WITH BICYCLIC CORE MOIETY PHENEX PHARMACEUTICALS AKTIENGESELLSCHAFT (DE) 2023-11-09 US disclosed
US-20230357214-A1 NOVEL LXR MODULATORS WITH BICYCLIC CORE MOIETY PHENEX PHARMACEUTICALS AKTIENGESELLSCHAFT (DE) 2023-11-09 US disclosed
CN-113666853-B Biaryl compounds useful as ROR gamma modulators 上海辉启生物医药科技有限公司 2023-04-18 CN disclosed
US-20220402867-A1 SULFO-SUBSTITUTED BIARYL COMPOUND OR SALT THEREOF, PREPARATION METHOD THEREFOR, AND USE THEREOF SHANGHAI LITEDD CO., LTD. (CN) 2022-12-22 US disclosed
US-20220402867-A1 SULFO-SUBSTITUTED BIARYL COMPOUND OR SALT THEREOF, PREPARATION METHOD THEREFOR, AND USE THEREOF SHANGHAI LITEDD CO., LTD. (CN) 2022-12-22 US disclosed
EP-4039674-A1 SULFO-SUBSTITUTED BIARYL COMPOUND OR SALT THEREOF, PREPARATION METHOD THEREFOR, AND USE THEREOF Shanghai Litedd Co., Ltd. (CN) 2022-08-10 EP disclosed
US-11364220-B2 Compounds and methods for inhibiting CPY26 enzymes QUEEN'S UNIVERSITY AT KINGSTON (CA) 2022-06-21 US disclosed
CN-112851557-B Sulfo-substituted biaryl compound or salt thereof, and preparation method and application thereof 上海辉启生物医药科技有限公司 2022-06-10 CN disclosed
CN-114502532-A Sulfo-substituted biaryl compound or salt thereof, and preparation method and application thereof 上海辉启生物医药科技有限公司 2022-05-13 CN disclosed
CN-109651208-B N-aryl sulfonamide compound, pharmaceutical composition and application thereof 中国科学院上海药物研究所 2022-01-04 CN disclosed
US-20090274632-A1 Identification of human T2R receptors that respond to bitter compounds that elicit the bitter taste in compositions, and the use thereof in assays to identify compounds that inhibit (block) bitter taste in composition and use thereof SENOMYX, INC. (US) 2009-11-05 US disclosed
CN-101443348-A Compounds and compositions as channel activating protease inhibitors IRM LLC (BM) 2009-05-27 CN disclosed
US-20090088368-A1 COMPOSITIONS COMPRISING THEM AS PPAR MODULATORS IRM LLC (BM) 2009-04-02 US disclosed
US-20090088368-A1 COMPOSITIONS COMPRISING THEM AS PPAR MODULATORS IRM LLC (BM) 2009-04-02 US disclosed
WO-2009025793-A2 HUMAN T2R BITTERNESS RECEPTORS AND USES THEREOF SENOMYX, INC. (US) 2009-02-26 WO disclosed
EP-2019837-A1 COMPOUNDS AND COMPOSITIONS AS CHANNEL ACTIVATING PROTEASE INHIBITORS IRM LLC (BM) 2009-02-04 EP disclosed
WO-2007140117-A1 COMPOUNDS AND COMPOSITIONS AS CHANNEL ACTIVATING PROTEASE INHIBITORS IRM LLC (BM) 2007-12-06 WO disclosed
US-20070276002-A1 Compounds and Compositions as Channel Activating Protease Inhibitors IRM LLC (BM) 2007-11-29 US disclosed
US-20070276002-A1 Compounds and Compositions as Channel Activating Protease Inhibitors IRM LLC (BM) 2007-11-29 US disclosed
US-20070276002-A1 Compounds and Compositions as Channel Activating Protease Inhibitors IRM LLC (BM) 2007-11-29 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (6 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090274632-A1 Identification of human T2R receptors that respond to bitter compounds that elicit the bitter taste in compositions, and the use thereof in assays to identify compounds that inhibit (block) bitter taste in composition and use thereof TAS2R50, TAS2R1, TAS2R30 CYP4F2 938/4885CYP4A11 2225/4885MMP9 4736/4885
US-20220402867-A1 SULFO-SUBSTITUTED BIARYL COMPOUND OR SALT THEREOF, PREPARATION METHOD THEREFOR, AND USE THEREOF RORB, RORA, RORC CYP4F2 132/4885CYP4A11 7/4885MMP9 3961/4885
US-20070276002-A1 Compounds and Compositions as Channel Activating Protease Inhibitors PRSS1, PRSS8, PRSS2 CYP4F2 4061/4885CYP4A11 3313/4885MMP9 140/4885
US-11364220-B2 Compounds and methods for inhibiting CPY26 enzymes CYP2A6, CYP27A1, CYP26B1 CYP4F2 23/4885CYP4A11 59/4885MMP9 3394/4885
US-20230357214-A1 NOVEL LXR MODULATORS WITH BICYCLIC CORE MOIETY NR1H2, NR1H3, NR1H4 CYP4F2 1149/4885CYP4A11 122/4885MMP9 4476/4885
US-20090088368-A1 COMPOSITIONS COMPRISING THEM AS PPAR MODULATORS PPARG, PPARA, PPARD CYP4F2 1420/4885CYP4A11 923/4885MMP9 2424/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.