SCHEMBL257394

SCHEMBL257394

Nc1nc(-c2ccccc2Cl)c(C(=O)c2cccc(Cl)c2)s1

nearest known ligand 0.61

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
RORB Q92753 8/20 0.61
GSK3B P49841 4/20 0.54
ADORA2A P29274 2/20 0.53
ADORA1 P30542 1/20 0.53
CCNA2 P20248 2/20 0.51
CDK2 P24941 2/20 0.51
ALDH1A1 P00352 1/20 0.47
RORC P51449 1/20 0.47
MAOB P27338 1/20 0.46
MYC P01106 1/20 0.43
WDR5 P61964 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL178186 0.89 RORB (0.54) RORBGSK3BADORA2AADORA1CCNA2
SCHEMBL257613 0.86 RORB (0.52) RORBADORA2AADORA1ALDH1A1RORC
SCHEMBL10092883 0.85 RORB (0.67) RORBADORA2AADORA1CCNA2CDK2
SCHEMBL257615 0.84 RORB (0.72) RORBADORA2ACCNA2CDK2ALDH1A1
SCHEMBL257393 0.82 RORB (0.60) RORBADORA2AADORA1CCNA2CDK2
SCHEMBL257203 0.81 RORB (0.67) RORBALDH1A1RORCMYCWDR5
SCHEMBL257432 0.80 RORB (0.74) RORBADORA2AADORA1CCNA2CDK2
SCHEMBL11274884 0.79 MYC (0.51) RORBALDH1A1RORCMYCWDR5
SCHEMBL2489836 0.79 MYC (0.51) RORBCDK2ALDH1A1RORCMYC
SCHEMBL30395217 0.79 MYC (0.51) RORBALDH1A1RORCMYCWDR5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012027965-A1 NOVEL COMPOUNDS GLAXO GROUP LIMITED (GB) 2012-03-08 WO disclosed