SCHEMBL257393

SCHEMBL257393

Nc1nc(-c2ccc(Cl)cc2)c(C(=O)c2cccc(Cl)c2)s1

nearest known ligand 0.60

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
RORB Q92753 9/20 0.60
CCNA2 P20248 2/20 0.50
CDK2 P24941 2/20 0.50
ALDH1A1 P00352 2/20 0.49
ADORA2A P29274 2/20 0.48
ADORA3 P0DMS8 1/20 0.48
ADORA1 P30542 1/20 0.48
POLB P06746 1/20 0.47
MEN1 O00255 1/20 0.47
MAPT P10636 1/20 0.47
KMT2A Q03164 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
L3MBTL1 Q9Y468 1/20 0.47
RORC P51449 1/20 0.46
MAOB P27338 1/20 0.45
CDK5 Q00535 2/20 0.45
CDK5R1 Q15078 2/20 0.45
LMNA P02545 1/20 0.44
NPSR1 Q6W5P4 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10092883 0.92 RORB (0.67) RORBCCNA2CDK2ALDH1A1ADORA2A
SCHEMBL257615 0.91 RORB (0.72) RORBCCNA2CDK2ALDH1A1ADORA2A
SCHEMBL178204 0.89 CDK5 (0.58) RORBCCNA2CDK2ADORA2AADORA3
SCHEMBL178218 0.88 ADORA3 (0.60) RORBALDH1A1ADORA2AADORA3ADORA1
SCHEMBL10092885 0.87 RORB (0.70) RORBADORA2AADORA3ADORA1MAPT
SCHEMBL257438 0.86 ADORA3 (0.54) RORBALDH1A1ADORA2AADORA3ADORA1
SCHEMBL257432 0.85 RORB (0.74) RORBCCNA2CDK2ALDH1A1ADORA2A
SCHEMBL10092890 0.83 RORB (0.65) RORBCCNA2CDK2RORCCDK5
SCHEMBL257616 0.83 ADORA3 (0.64) RORBALDH1A1ADORA2AADORA3ADORA1
SCHEMBL257394 0.82 RORB (0.61) RORBCCNA2CDK2ALDH1A1ADORA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012027965-A1 NOVEL COMPOUNDS GLAXO GROUP LIMITED (GB) 2012-03-08 WO disclosed