SCHEMBL2575382

SCHEMBL2575382

CC1(C)Cc2cc(C(=O)O)ccc2NC1c1cccc(NCCCc2ccccc2)c1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CSNK2A2 P19784 1/20 0.37
CSNK2B P67870 1/20 0.37
CSNK2A1 P68400 1/20 0.37
NR1H4 Q96RI1 1/20 0.36
ITGB3 P05106 1/20 0.36
ITGAV P06756 1/20 0.36
HDAC1 Q13547 1/20 0.36
HDAC8 Q9BY41 1/20 0.36
HDAC6 Q9UBN7 1/20 0.36
BRAF P15056 1/20 0.35
KDM4E B2RXH2 2/20 0.35
EPHX1 P07099 1/20 0.35
KMT2A Q03164 5/20 0.35
MEN1 O00255 3/20 0.35
LMNA P02545 3/20 0.35
ALDH1A1 P00352 2/20 0.35
HTT P42858 2/20 0.35
SMN1; SMN2 Q16637 2/20 0.35
PIK3CD O00329 1/20 0.35
TP53 P04637 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2568247 0.92 HTR7 (0.42) KMT2AMEN1LMNAALDH1A1SMN1; SMN2
SCHEMBL2530664 0.86 GAA (0.47) ALDH1A1HTTMAPTNPC1RAB9A
SCHEMBL2532947 0.84 RAB9A (0.44) KMT2AMEN1SMN1; SMN2TP53MAPT
SCHEMBL2530890 0.84 KMT2A (0.43) KDM4EKMT2AMEN1LMNAALDH1A1
SCHEMBL2527836 0.82 F10 (0.40) ALDH1A1SMN1; SMN2TP53RAB9AGAA
SCHEMBL12219890 0.81 KMO (0.43) KDM4EKMT2AMEN1ALDH1A1HTT
SCHEMBL2535130 0.81 KMT2A (0.46) NR1H4KMT2AMEN1TP53POLB
SCHEMBL2532410 0.81 NR4A1 (0.33) ITGB3ITGAVKDM4EKMT2AMEN1
SCHEMBL2530126 0.80 ALDH1A1 (0.40) KDM4EKMT2AMEN1ALDH1A1MAPT
SCHEMBL2531699 0.80 KDM1A (0.47) NR1H4HDAC1HDAC8HDAC6KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2558449-A1 NOVEL 3,3-DIMETHYL TETRAHYDROQUINOLINE DERIVATIVES F. Hoffmann-La Roche AG (CH) 2013-02-20 EP disclosed
WO-2011128251-A1 NOVEL 3,3-DIMETHYL TETRAHYDROQUINOLINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2011-10-20 WO disclosed