SCHEMBL25754916

SCHEMBL25754916

FC(F)(F)c1cnc(-c2ccc(Cl)cc2)[nH]1

nearest known ligand 0.67

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
SCN2A Q99250 3/20 0.51
DGAT1 O75907 9/20 0.49
NPY5R Q15761 1/20 0.43
TRPV1 Q8NER1 1/20 0.43
COMT P21964 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17868458 0.84 DGAT1 (0.50) SCN2ADGAT1TRPV1COMT
SCHEMBL11260682 0.82 DGAT1 (0.40) SCN2ADGAT1
SCHEMBL17678002 0.82 DGAT1 (0.49) SCN2ADGAT1TRPV1COMT
SCHEMBL17868402 0.82 DGAT1 (0.53) SCN2ADGAT1
SCHEMBL9940238 0.82 TRPV1 (0.62) SCN2ADGAT1TRPV1COMT
SCHEMBL3584568 0.81 SCN2A (0.58) SCN2ADGAT1NPY5R
SCHEMBL11245211 0.80 HRH1 (0.56) SCN2ANPY5R
SCHEMBL12499046 0.79 DGAT1 (0.46) SCN2ADGAT1TRPV1COMT
SCHEMBL23847030 0.78 DGAT1 (0.59) SCN2ADGAT1
SCHEMBL18865669 0.78 DGAT1 (0.49) SCN2ADGAT1NPY5R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4727549-A2 PLASMODIUM FALCIPARUM BLOOD STAGE INHIBITORS University of Georgia Research Foundation, Inc. (US) 2026-04-22 EP disclosed
US-20260097046-A1 PLASMODIUM FALCIPARUM BLOOD STAGE INHIBITORS UNIV GEORGIA (US) 2026-04-09 US disclosed
WO-2024258900-A2 PLASMODIUM FALCIPARUM BLOOD STAGE INHIBITORS UNIVERSITY OF GEORGIA RESEARCH FOUNDATION, INC. (US) 2024-12-19 WO disclosed
US-20230174523-A1 BENZENESULFONAMIDE DERIVATIVES AS TRAP1 MODULATORS AND USES THEREOF AMATHUS THERAPEUTICS, INC. (US) 2023-06-08 US disclosed
US-20230174523-A1 BENZENESULFONAMIDE DERIVATIVES AS TRAP1 MODULATORS AND USES THEREOF AMATHUS THERAPEUTICS, INC. (US) 2023-06-08 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230174523-A1 BENZENESULFONAMIDE DERIVATIVES AS TRAP1 MODULATORS AND USES THEREOF TRAP1, PINK1, TP53BP1 SCN2A 818/4885DGAT1 3633/4885NPY5R 3221/4885
US-20260097046-A1 PLASMODIUM FALCIPARUM BLOOD STAGE INHIBITORS SUB1, PFN1, HCCS SCN2A 2686/4885DGAT1 1115/4885NPY5R 2804/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.